General method for synthesis of 2-heterocyclic N-methyliminodiacetic acid boronates

Graham R. Dick; David M. Knapp; Eric P. Gillis; Martin D. Burke

doi:10.1021/ol100671v

General method for synthesis of 2-heterocyclic N-methyliminodiacetic acid boronates

Graham R. Dick, David M. Knapp, Eric P. Gillis, Martin D. Burke

Research output: Contribution to journal › Article › peer-review

Abstract

A wide range of 2-pyridyl and other difficult-to-access heterocyclic N-methyliminodiacetic acid boronates can be readily prepared from the corresponding bromides via a new method involving direct transligation of 2-heterocyclic trialkoxyborate salts with N-methyliminodiacetic acid (MIDA) at elevated temperatures.

Original language	English (US)
Pages (from-to)	2314-2317
Number of pages	4
Journal	Organic Letters
Volume	12
Issue number	10
DOIs	https://doi.org/10.1021/ol100671v
State	Published - May 21 2010

ASJC Scopus subject areas

Biochemistry
Physical and Theoretical Chemistry
Organic Chemistry

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10.1021/ol100671v

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abstract = "A wide range of 2-pyridyl and other difficult-to-access heterocyclic N-methyliminodiacetic acid boronates can be readily prepared from the corresponding bromides via a new method involving direct transligation of 2-heterocyclic trialkoxyborate salts with N-methyliminodiacetic acid (MIDA) at elevated temperatures.",

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AU - Gillis, Eric P.

AU - Burke, Martin D.

PY - 2010/5/21

Y1 - 2010/5/21

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AB - A wide range of 2-pyridyl and other difficult-to-access heterocyclic N-methyliminodiacetic acid boronates can be readily prepared from the corresponding bromides via a new method involving direct transligation of 2-heterocyclic trialkoxyborate salts with N-methyliminodiacetic acid (MIDA) at elevated temperatures.

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General method for synthesis of 2-heterocyclic N-methyliminodiacetic acid boronates

Abstract

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