Provided are methods for site- and stereo-retentive cross-couplings with unactivated secondary boronic acids, which methods are particularly useful in building block-based approach for small molecule synthesis. Also provided is a method of forming an air-stable chiral secondary boronic acid.
Original languageEnglish (US)
U.S. patent number10072028
Filing date11/3/14
StatePublished - Sep 11 2018


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