Abstract
Provided are methods for site- and stereo-retentive cross-couplings with unactivated secondary boronic acids, which methods are particularly useful in building block-based approach for small molecule synthesis. Also provided is a method of forming an air-stable chiral secondary boronic acid.
| Original language | English (US) |
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| U.S. patent number | 10072028 |
| Filing date | 11/3/14 |
| State | Published - Sep 11 2018 |