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  A mutant form of ERα associated with estrogen insensitivity affects the coupling between ligand binding and coactivator recruitment

  Li, Y., Coons, L. A., Houtman, R., Carlson, K. E., Martin, T. A., Mayne, C. G., Melchers, D., Jefferson, T. B., Ramsey, J. T., Katzenellenbogen, J. A. & Korach, K. S., Sep 22 2020, In: Science Signaling. 13, 650, eaaw4653.

  Research output: Contribution to journal › Article › peer-review

  • Estrogen Receptors
  • Estrogens
  • Ligands
  • Missense Mutation
  • Gene encoding

• Cyclic Ketoximes as Estrogen Receptor β Selective Agonists

  Granchi, C., Lapillo, M., Spena, C. R., Rizzolio, F., Tuccinardi, T., Martin, T. A., Carlson, K. E., Katzenellenbogen, J. A. & Minutolo, F., 2016, In: ChemMedChem. p. 1752-1761 10 p.

  Research output: Contribution to journal › Article › peer-review

  • Oximes
  • Estrogen Receptors
  • Estrogens
  • salicylaldoxime
  • Molecular modeling

• Estrogen receptor alpha somatic mutations Y537S and D538G confer breast cancer endocrine resistance by stabilizing the activating function-2 binding conformation

  Fanning, S. W., Mayne, C. G., Dharmarajan, V., Carlson, K. E., Martin, T. A., Novick, S. J., Toy, W., Green, B., Panchamukhi, S., Katzenellenbogen, B. S., Tajkhorshid, E., Griffin, P. R., Shen, Y., Chandarlapaty, S., Katzenellenbogen, J. A. & Greene, G. L., Feb 2 2016, In: eLife. 5, FEBRUARY2016, e12792.

  Research output: Contribution to journal › Article › peer-review

  • Conformations
  • Estrogen Receptor alpha
  • Estrogen Receptor Modulators
  • Breast Neoplasms
  • Mutation

• Licorice root components in dietary supplements are selective estrogen receptor modulators with a spectrum of estrogenic and anti-estrogenic activities

  Boonmuen, N., Gong, P., Ali, Z., Chittiboyina, A. G., Khan, I., Doerge, D. R., Helferich, W. G., Carlson, K. E., Martin, T., Piyachaturawat, P., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 2016, In: Steroids. 105, p. 42-49 8 p.

  Research output: Contribution to journal › Article › peer-review

  • Dietary supplements
  • liquiritigenin
  • isoliquiritigenin
  • Glycyrrhiza
  • Selective Estrogen Receptor Modulators

• Reconstruction of Lead Acid Battery Negative Electrodes after Hard Sulfation Using Controlled Chelation Chemistry

  Gossage, Z. T., Guo, F., Hatfield, K. O., Martin, T. A., Tian, Q., Gao, E. J., Kumar, A., Rodríguez-López, J. & Zhao, H., Jan 9 2020, In: Journal of the Electrochemical Society. 167, 12, 120537.

  Research output: Contribution to journal › Article › peer-review

  • Chelation
  • Lead acid batteries
  • Ethylenediaminetetraacetic acid
  • Edetic Acid
  • Electrodeposition

• Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer

  Xiong, R., Patel, H. K., Gutgesell, L. M., Zhao, J., Delgado-Rivera, L., Pham, T. N. D., Zhao, H., Carlson, K., Martin, T., Katzenellenbogen, J. A., Moore, T. W., Tonetti, D. A. & Thatcher, G. R. J., Jan 14 2016, In: Journal of Medicinal Chemistry. 59, 1, p. 219-237 19 p.

  Research output: Contribution to journal › Article › peer-review

  • Tamoxifen
  • Estrogens
  • Breast Neoplasms
  • Estrogen Receptors
  • benzothiophene

• The SERM/SERD bazedoxifene disrupts ESR1 helix 12 to overcome acquired hormone resistance in breast cancer cells

  Fanning, S. W., Jeselsohn, R., Dharmarajan, V., Mayne, C. G., Karimi, M., Buchwalter, G., Houtman, R., Toy, W., Fowler, C. E., Han, R., Lainé, M., Carlson, K. E., Martin, T. A., Nowak, J., Nwachukwu, J. C., Hosfield, D. J., Chandarlapaty, S., Tajkhorshid, E., Nettles, K. W., Griffin, P. R. & 4 others, Shen, Y., Katzenellenbogen, J. A., Brown, M. & Greene, G. L., Nov 1 2018, In: eLife. 7, e37161.

  Research output: Contribution to journal › Article › peer-review

  • bazedoxifene
  • Selective Estrogen Receptor Modulators
  • Estrogen Receptor Modulators
  • Estrogen Receptor alpha
  • Tamoxifen