Benita S Katzenellenbogen

1970 …2020
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Research Output 1970 2020

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Estrogen receptors α and β as determinants of gene expression: Influence of ligand, dose, and chromatin binding

Chang, E. C., Charn, T. H., Park, S. H., Helferich, W. G., Komm, B., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., May 1 2008, In : Molecular Endocrinology. 22, 5, p. 1032-1043 12 p.

Research output: Contribution to journalArticle

Genistein
Estrogen Receptors
Chromatin
Ligands
Gene Expression

Estrogen receptor transformation in MCF-7 breast cancer cells: Characterization by immunochemical and sedimentation analyses

Miller, M. A., Greene, G. L. & Katzenellenbogen, B. S., Jan 1 1984, In : Endocrinology. 114, 1, p. 296-298 3 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Breast Neoplasms
Buffers
Sucrose
MCF-7 Cells
Aryl Hydrocarbon Receptors
Estrogen Receptors
Estrogens
Gene expression
Crosstalk

Estrogen receptor β ligands: Recent advances and biomedical applications

Minutolo, F., Macchia, M., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., May 1 2011, In : Medicinal Research Reviews. 31, 3, p. 364-442 79 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Ligands
Non-Steroidal Estrogens
Therapeutic Uses
Endometriosis
Estrogen Receptors
Apoptosis
Breast Neoplasms
Gene Expression
Histones

Estrogen receptor-β potency-selective ligands: Structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues

Meyers, M. J., Sun, J., Carlson, K. E., Marriner, G. A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Nov 22 2001, In : Journal of Medicinal Chemistry. 44, 24, p. 4230-4251 22 p.

Research output: Contribution to journalArticle

Acetylene
Estrogen Receptor alpha
Structure-Activity Relationship
Estrogen Receptors
Ligands

Estrogen-regulated gene networks in human breast cancer cells: Involvement of E2F1 in the regulation of cell proliferation

Stender, J. D., Frasor, J., Komm, B., Chang, K. C. N., Kraus, W. L. & Katzenellenbogen, B. S., Sep 1 2007, In : Molecular Endocrinology. 21, 9, p. 2112-2123 12 p.

Research output: Contribution to journalArticle

Gene Regulatory Networks
Estrogens
Cell Proliferation
Breast Neoplasms
Estrogen Receptors

Estrogen-regulated prohibitin is required for mouse uterine development and adult function

He, B., Kim, T. H., Kommagani, R., Feng, Q., Lanz, R. B., Jeong, J. W., DeMayo, F. J., Katzenellenbogen, B. S., Lydon, J. P. & O'Malley, B. W., Mar 1 2011, In : Endocrinology. 152, 3, p. 1047-1056 10 p.

Research output: Contribution to journalArticle

Estrogens
Estrogen Receptors
Uterus
Steroid Receptors
Genes

Estrogen regulation of human osteoblast function is determined by the stage of differentiation and the estrogen receptor isoform

Waters, K. M., Rickard, D. J., Lawrence Riggs, B., Khosla, S., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Moore, J. & Spelsberg, T. C., Nov 13 2001, In : Journal of Cellular Biochemistry. 83, 3, p. 448-462 15 p.

Research output: Contribution to journalArticle

Osteoblasts
Estrogen Receptors
Tamoxifen
Protein Isoforms
Estrogens

Estrogen regulation of the glucuronidation enzyme UGT2B15 in estrogen receptor-positive breast cancer cells

Harrington, W. R., Sengupta, S. & Katzenellenbogen, B. S., Jul 24 2006, In : Endocrinology. 147, 8, p. 3843-3850 8 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Breast Neoplasms
Enzymes
Glucuronosyltransferase

Estrogens and androgens inhibit association of RANKL with the pre-osteoblast membrane through post-translational mechanisms

Martin, A., Yu, J., Xiong, J., Khalid, A. B., Katzenellenbogen, B., Kim, S. H., Katzenellenbogen, J. A., Malaivijitnond, S., Gabet, Y., Krum, S. A. & Frenkel, B., Dec 2017, In : Journal of Cellular Physiology. 232, 12, p. 3798-3807 10 p.

Research output: Contribution to journalArticle

Osteoblasts
Dihydrotestosterone
Androgens
Estrogens
Association reactions

Estrone interaction with the rat uterus: In vitro response and nuclear uptake

Ruh, T. S., Katzenellenbogen, B. S., Katzenellenbogen, J. A. & Gorski, J., Jan 1973, In : Endocrinology. 92, 1, p. 125-134 10 p.

Research output: Contribution to journalArticle

Estrone
Uterus
Estradiol
Estriol
Estrogens

Evaluation of wild yam (Dioscorea villosa) root extract as a potential epigenetic agent in breast cancer cells

Aumsuwan, P., Khan, S. I., Khan, I. A., Avula, B., Walker, L. A., Helferich, W. G., Katzenellenbogen, B. S. & Dasmahapatra, A. K., Jan 1 2014, In : In Vitro Cellular and Developmental Biology - Animal. 51, 1, p. 59-71 13 p.

Research output: Contribution to journalArticle

5-methyldeoxycytidine
Dioscorea
Epigenomics
MCF-7 Cells
Breast Neoplasms
Estrogen Receptor Modulators
Estrogen Receptors
Transcriptional Activation
Hormones
DNA
Gene Transfer Techniques
Estrogen Receptors
Genes
Cells
Hormones

Expression of steroid hormone receptors in BRCA1-associated ovarian carcinomas

Aghmesheh, M., Edwards, L., Clarke, C. L., Byth, K., Katzenellenbogen, B. S., Russell, P. J., Friedlander, M., Tucker, K. M. & De Fazio, A., Apr 2005, In : Gynecologic Oncology. 97, 1, p. 16-25 10 p.

Research output: Contribution to journalArticle

Steroid Receptors
Estrogen Receptors
Ovarian Neoplasms
Hormones
Carcinoma

Extranuclear estrogen receptor-α stimulates NeuroD1 binding to the insulin promoter and favors insulin synthesis

Wong, W. P. S., Tiano, J. P., Liu, S., Hewitt, S. C., Le May, C., Dalle, S., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Korach, K. S. & Mauvais-Jarvis, F., Jul 20 2010, In : Proceedings of the National Academy of Sciences of the United States of America. 107, 29, p. 13057-13062 6 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Insulin
Response Elements
Islets of Langerhans
Estrogens
Non-Steroidal Estrogens
Estrogen Receptor Modulators
Isomerization
Isomers
Estrogen Receptors

Full antagonism of the estrogen receptor without a prototypical ligand side chain

Srinivasan, S., Nwachukwu, J. C., Bruno, N. E., Dharmarajan, V., Goswami, D., Kastrati, I., Novick, S., Nowak, J., Cavett, V., Zhou, H. B., Boonmuen, N., Zhao, Y., Min, J., Frasor, J., Katzenellenbogen, B. S., Griffin, P. R., Katzenellenbogen, J. A. & Nettles, K. W., Jan 1 2017, In : Nature chemical biology. 13, 1, p. 111-118 8 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Ligands
Breast Neoplasms
Chemoprevention
Therapeutic Uses

Fundamental differences in the action of estrogens and antiestrogens on the uterus: comparison between compounds with similar duration of action

Katzenellenbogen, B. S., Ferguson, E. R., Lan, N. C., Ferguson, E. R. & Lan, N. C., May 1977, In : Endocrinology. 100, 5, p. 1252-1259 8 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Cytoplasmic and Nuclear Receptors
Uterus
Estrogens
Estradiol

Furans with basic side chains: Synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha

Mortensen, D. S., Rodriguez, A. L., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Sep 17 2001, In : Bioorganic and Medicinal Chemistry Letters. 11, 18, p. 2521-2524 4 p.

Research output: Contribution to journalArticle

Furans
Estrogen Receptor alpha
Phenol
Estrogen Receptors
Ligands

Gene expression preferentially regulated by tamoxifen in breast cancer cells and correlations with clinical outcome

Frasor, J., Chang, E. C., Komm, B., Lin, C. Y., Vega, V. B., Liu, E. T., Miller, L. D., Smeds, J., Bergh, J. & Katzenellenbogen, B. S., Jul 15 2006, In : Cancer Research. 66, 14, p. 7334-7340 7 p.

Research output: Contribution to journalArticle

Tamoxifen
Breast Neoplasms
Gene Expression
Estrogen Receptors
Genes

General esterases of silkmoth moulting fluid: Preliminary characterization

Katzenellenbogen, B. S. & Kafatos, F. C., Jun 1971, In : Journal of insect physiology. 17, 6

Research output: Contribution to journalArticle

Molting
Bombyx
Esterases
esterases
molting

Genetic deletion of the repressor of estrogen receptor activity (REA) enhances the response to estrogen in target tissues in vivo

Park, S. E., Xu, J., Frolova, A., Liao, L., O'Malley, B. W. & Katzenellenbogen, B. S., Mar 1 2005, In : Molecular and cellular biology. 25, 5, p. 1989-1999 11 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Uterus
Wild Animals
Genes

Genome-wide analysis of estrogen receptor α DNA binding and tethering mechanisms identifies Runx1 as a novel tethering factor in receptor-mediated transcriptional activation

Stender, J. D., Kim, K., Charn, T. H., Komm, B., Chang, K. C. N., Kraus, W. L., Benner, C., Glass, C. K. & Katzenellenbogen, B. S., Aug 1 2010, In : Molecular and cellular biology. 30, 16, p. 3943-3955 13 p.

Research output: Contribution to journalArticle

Estrogen Receptor alpha
Estrogen Receptors
Transcriptional Activation
Genome
Response Elements

Genome-wide dynamics of chromatin binding of estrogen receptors α and β: Mutual restriction and competitive site selection

Charn, T. H., Liu, E. T. B., Chang, E. C., Lee, Y. K., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 2010, In : Molecular Endocrinology. 24, 1, p. 47-59 13 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Chromatin
Binding Sites
Genome
Cytoplasmic and Nuclear Receptors
Mitogen-Activated Protein Kinase 1
Estrogen Receptors
Genes
Cytoplasmic and Nuclear Receptors
Mitogen-Activated Protein Kinases

Haploinsufficiency of the corepressor of estrogen receptor activity (REA) enhances estrogen receptor function in the mammary gland

Mussi, P., Liao, L., Park, S. E., Ciana, P., Maggi, A., Katzenellenbogen, B. S., Xu, J. & O'Malley, B. W., Nov 7 2006, In : Proceedings of the National Academy of Sciences of the United States of America. 103, 45, p. 16716-16721 6 p.

Research output: Contribution to journalArticle

Haploinsufficiency
Co-Repressor Proteins
Human Mammary Glands
Estrogen Receptors
Estrogens

Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model

Paterni, I., Bertini, S., Granchi, C., Tuccinardi, T., Macchia, M., Martinelli, A., Caligiuri, I., Toffoli, G., Rizzolio, F., Carlson, K. E., Katzenellenbogen, B. S., Katzenellenbogen, J. A. & Minutolo, F., Feb 12 2015, In : Journal of Medicinal Chemistry. 58, 3, p. 1184-1194 11 p.

Research output: Contribution to journalArticle

Glioma
Estrogen Receptors
Estrogens
Heterografts
Pharmacology

Highly sensitive quantitative imaging for monitoring single cancer cell growth kinetics and drug response

Mir, M., Bergamaschi, A., Katzenellenbogen, B. S. & Popescu, G., Feb 18 2014, In : PloS one. 9, 2, e89000.

Research output: Contribution to journalArticle

Light interference
Growth kinetics
Cell growth
cell growth
Microscopic examination

Hormonal Modulation of HER-2/neu Protooncogene Messenger Ribonucleic Acid and pl85 Protein Expression in Human Breast Cancer Cell Lines

Read, L. D., Keith, D., Slamon, D. J. & Katzenellenbogen, B. S., Jul 1 1990, In : Cancer Research. 50, 13, p. 3947-3951 5 p.

Research output: Contribution to journalArticle

RNA
Breast Neoplasms
Cell Line
Messenger RNA
Progestins

Hormone binding and transcription activation by estrogen receptors: Analyses using mammalian and yeast systems

Katzenellenbogen, B. S., Bhardwaj, B., Fang, H., Ince, B. A., Pakde, F., Reese, J. C., Schodin, D. & Wrenn, C. K., Dec 1993, In : Journal of Steroid Biochemistry and Molecular Biology. 47, 1-6, p. 39-48 10 p.

Research output: Contribution to journalArticle

Transcription
Estrogen Receptors
Yeast
Transcriptional Activation
Yeasts
Granulosa Cells
Progesterone Receptors
Genetic Promoter Regions
Cyclic AMP
Estradiol

Human endometrial cells in primary tissue culture: Modulation of progesterone receptor level by estrogens in vitro

Eckert, R. L. & Katzenellenbogen, B. S., Jan 1 1980, In : Biology of reproduction. 22, SUPPL. 1, p. No. 160

Research output: Contribution to journalArticle

Progesterone Receptors
Estrogens
In Vitro Techniques
Tissue culture
Diethylstilbestrol
Cell proliferation
Estrogens
Cell Proliferation
Estradiol Congeners
Tissue culture
Progesterone Receptors
Zeranol
Estradiol
Estrogen Receptor beta
Monoclonal Antibodies
Tissue
Antibodies
Granulosa Cells
Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Ligands
Estradiol

Human estrogen receptor mutants with altered estrogen and antiestrogen ligand discrimination

Pakdel, F. & Katzenellenbogen, B. S., Jan 1 1992, In : Journal of Biological Chemistry. 267, 5, p. 3429-3437 9 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Ligands
Amino Acids

Identification of amino acids in the hormone binding domain of the human estrogen receptor important in estrogen binding

Ekena, K., Weis, K. E., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Sep 5 1996, In : Journal of Biological Chemistry. 271, 33, p. 20053-20059 7 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Hormones
Ligands
Amino Acids
Estrogens
Hormones
Genes
Progesterone Receptors
Estrogen Receptors
Estrogen Receptors
Estrogens
Hormones
Estrogen Receptor Modulators
Steroid Receptors

Identification of cysteine 530 as the covalent attachment site of an affinity-labeling estrogen (ketononestrol aziridine) and antiestrogen (tamoxifen aziridine) in the human estrogen receptor

Harlow, K. W., Smith, D. N., Katzenellenbogen, J. A., Greene, G. L. & Katzenellenbogen, B. S., 1989, In : Journal of Biological Chemistry. 264, 29, p. 17476-17485 10 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Labeling
Cysteine
Estrogens

Identification of multiple, widely spaced estrogen-responsive regions in the rat progesterone receptor gene

Kraus, W. L., Montano, M. M. & Katzenellenbogen, B. S., Aug 1 1994, In : Molecular Endocrinology. 8, 8, p. 952-969 18 p.

Research output: Contribution to journalArticle

Progesterone Receptors
Estrogens
Genes
Response Elements
Base Pairing
Estrogen Receptors
Transcriptional Activation
Cysteine
Ligands
Estrogen Receptor Modulators

Impact of estrogen receptor β on gene networks regulated by estrogen receptor α in breast cancer cells

Chang, E. C., Frasor, J., Komm, B. & Katzenellenbogen, B. S., Sep 22 2006, In : Endocrinology. 147, 10, p. 4831-4842 12 p.

Research output: Contribution to journalArticle

Gene Regulatory Networks
Estrogen Receptors
Breast Neoplasms
Gene Expression
Genes

Inactive proteinases in silkmoth moulting gel

Katzenellenbogen, B. S. & Kafatos, F. C., May 1971, In : Journal of insect physiology. 17, 5, p. 823-832 10 p.

Research output: Contribution to journalArticle

Molting
Bombyx
molting
Peptide Hydrolases
proteinases

Indazole estrogens: Highly selective ligands for the estrogen receptor β

De Angelis, M., Stossi, F., Carlson, K. A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Feb 24 2005, In : Journal of Medicinal Chemistry. 48, 4, p. 1132-1144 13 p.

Research output: Contribution to journalArticle

Indazoles
Estrogen Receptors
Estradiol
Estrogens
Ligands
Steroid Receptors
Progesterone Receptors
Estrogen Receptors
Hormones
Ligands

In memoriam: Jack Gorski (1931-2006).

Katzenellenbogen, B. S., Nov 2006, In : Molecular endocrinology (Baltimore, Md.). 20, 11, p. 2611-2612 2 p.

Research output: Contribution to journalArticle

21st Century History
20th Century History
Endocrinology