Benita S Katzenellenbogen

1970 …2019
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Research Output 1970 2019

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Article
Estrogen Receptor Modulators
Tritium
Estrogen Receptors
Propylene Glycols
Propylene Glycol
Estrogen Receptor Modulators
Estrogens
Molecular Weight
Breast Neoplasms
Proteins
Promegestone
Progestins
Progesterone Receptors
Cells
Breast Neoplasms
Estrogen Receptor Modulators
Estrogen Receptors
Breast Neoplasms
Neoplasms
Peroxidase

A repressive role for prohibitin in estrogen signaling

He, B., Feng, Q., Mukherjee, A., Lonard, D. M., DeMayo, F. J., Katzenellenbogen, B. S., Lydon, J. P. & O'Malley, B. W., Feb 1 2008, In : Molecular Endocrinology. 22, 2, p. 344-360 17 p.

Research output: Contribution to journalArticle

Estrogens
Co-Repressor Proteins
Estrogen Receptors
prohibitin
Protein Stability

A role for Akt in mediating the estrogenic functions of epidermal growth factor and insulin-like growth factor I

Martin, M. B., Franke, T. F., Stoica, G. E., Chambon, P., Katzenellenbogen, B. S., Stoica, B. A., McLemore, M. S., Olivo, S. E. & Stoica, A., Jan 1 2000, In : Endocrinology. 141, 12, p. 4503-4511 9 p.

Research output: Contribution to journalArticle

Insulin-Like Growth Factor I
Epidermal Growth Factor
Transfection
Phosphatidylinositol 3-Kinase
70-kDa Ribosomal Protein S6 Kinases
Nuclear Receptor Co-Repressor 1
Aryl Hydrocarbon Receptors
Gene expression
Estrogen Receptors
Chromatin

A transcriptionally active estrogen receptor mutant is a novel type of dominant negative inhibitor of estrogen action

McInerney, E. M., Ince, B. A., Shapiro, D. J. & Katzenellenbogen, B. S., Dec 17 1996, In : Molecular Endocrinology. 10, 12, p. 1519-1526 8 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Response Elements
DNA
Amino Acid Substitution

Bibenzyl- and stilbene-core compounds with non-polar linker atom substituents as selective ligands for estrogen receptor beta

Waibel, M., De Angelis, M., Stossi, F., Kieser, K. J., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Sep 1 2009, In : European Journal of Medicinal Chemistry. 44, 9, p. 3412-3424 13 p.

Research output: Contribution to journalArticle

Stilbenes
Estrogen Receptor beta
Estrogen Receptors
Ligands
Atoms

Bioactivities, Estrogen Receptor Interactions, and Plasminogen Activator-inducing Activities of Tamoxifen and Hydroxy-tamoxifen Isomers in MCF-7 Human Breast Cancer Cells

Katzenellenbogen, B. S., Norman, M. J., Eckert, R. L., Peltz, S. W. & Mangel, W. F., Jan 1 1984, In : Cancer Research. 44, 1, p. 112-119 8 p.

Research output: Contribution to journalArticle

Plasminogen Activators
Tamoxifen
Estrogen Receptors
Breast Neoplasms
Progesterone Receptors

Biological activities of tamoxifen aziridine, an antiestrogen-based affinity label for the estrogen receptor, in vivo and in vitro

Wei, L. L., Mangel, W. F. & Katzenellenbogen, B. S., Dec 1985, In : Journal of Steroid Biochemistry. 23, 6 PART 1, p. 875-881 7 p.

Research output: Contribution to journalArticle

Affinity Labels
Estrogen Receptor Modulators
Bioactivity
Estrogen Receptors
Tamoxifen

Biological Activity and Receptor Binding of a Strongly Interacting Estrogen in Human Breast Cancer Cells

Reiner, G. C. A., Katzenellenbogen, B. S., Bindal, R. D. & Katzenellenbogen, J. A., Jun 1 1984, In : Cancer Research. 44, 6, p. 2302-2308 7 p.

Research output: Contribution to journalArticle

Estradiol
Estrogens
Estrogen Receptors
Breast Neoplasms
MCF-7 Cells

Biological Potency and Uterine Estrogen Receptor Interactions of the Metabolites of the Antiestrogens CI628 and U23, 469

Hayes, J. R., Rorke, E. A., Robertson, D. W., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 1981, In : Endocrinology. 108, 1, p. 164-172 9 p.

Research output: Contribution to journalArticle

Nitromifene
Estrogen Receptor Modulators
Estrogen Receptors
Estradiol
Cytoplasmic and Nuclear Receptors

Biology and receptor interactions of estriol and estriol derivatives in vitro and in vivo

Katzenellenbogen, B. S., Apr 1984, In : Journal of Steroid Biochemistry. 20, 4 PART 2, p. 1033-1037 5 p.

Research output: Contribution to journalArticle

Estriol
Derivatives
Estrogens
Cell culture
Estrogen Receptors

Bivalent ligands as probes of estrogen receptor action

Bergmann, K. E., Wooge, C. H., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jun 1994, In : Journal of Steroid Biochemistry and Molecular Biology. 49, 2-3, p. 139-152 14 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Hexestrol
Ligands
Reporter Genes
Estrogen Antagonists

Bridged bicyclic cores containing a 1,1-diarylethylene motif are high-affinity subtype-selective ligands for the estrogen receptor

Muthyala, R. S., Sheng, S., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Apr 24 2003, In : Journal of Medicinal Chemistry. 46, 9, p. 1589-1602 14 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Ligands
Estrogens
Non-Steroidal Estrogens
Terpenes

Caveolin-1 potentiates estrogen receptor α (ERα) signaling. Caveolin-1 drives ligand-independent nuclear translocation and activation of ERα

Schlegel, A., Wang, C., Katzenellenbogen, B. S., Pestell, R. G. & Lisanti, M. P., Nov 19 1999, In : Journal of Biological Chemistry. 274, 47, p. 33551-33556 6 p.

Research output: Contribution to journalArticle

Caveolin 1
Estrogen Receptors
Chemical activation
Ligands
Signal transduction
Estrogen Receptor Modulators
Estrogen Receptors
Binding Sites
Breast Neoplasms
Cell Line

Characterization and regulation of estrogen and progesterone receptors in breast cancer.

Read, L. D. & Katzenellenbogen, B. S., Dec 1 1992, In : Cancer treatment and research. 61, p. 277-299 23 p.

Research output: Contribution to journalArticle

Neoplastic Gene Expression Regulation
Hormone-Dependent Neoplasms
Neoplasm Proteins
Growth Substances
Progestins
Cell Extracts
Estrogen Receptors
Transcriptional Activation
Chemical activation
Hormones
Progesterone Receptors
Estrogen Receptors
Estrogens
Breast Neoplasms
Growth

Characterization of the biological roles of the estrogen receptors, ERα and ERβ, in estrogen target tissues in vivo through the use of an ERα-selective ligand

Harris, H. A., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Nov 1 2002, In : Endocrinology. 143, 11, p. 4172-4177 6 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Ligands
Arcuate Nucleus of Hypothalamus
Complement C3

Characterization of the estrogen receptor and its dynamics in MCF-7 human breast cancer cells using a covalently attaching antiestrogen

Monsma, F. J., Katzenellenbogen, B. S., Miller, M. A., Ziegler, Y. S. & Katzenellenbogen, J. A., Jan 1 1984, In : Endocrinology. 115, 1, p. 143-153 11 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Cytoplasmic and Nuclear Receptors
Breast Neoplasms
Sodium Dodecyl Sulfate

Characterization of the interactions of estrogen receptor and MNAR in the activation of cSrc

Barletta, F., Wong, C. W., McNally, C., Komm, B. S., Katzenellenbogen, B. S. & Cheskis, B. J., May 1 2004, In : Molecular Endocrinology. 18, 5, p. 1096-1108 13 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
src Homology Domains
Phosphotyrosine
Mutation

Characterization of the pharmacophore properties of novel selective estrogen receptor downregulators (SERDs)

Kieser, K. J., Kim, D. W., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Apr 22 2010, In : Journal of Medicinal Chemistry. 53, 8, p. 3320-3329 10 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Ligands
Cyclofenil
Ether
Hormones

Characterization of the subunit nature of nuclear estrogen receptors by chemical cross-linking and dense amino acid labeling

Miller, M. A., Mullick, A., Greene, G. L. & Katzenellenbogen, B. S., Aug 1985, In : Endocrinology. 117, 2, p. 515-522 8 p.

Research output: Contribution to journalArticle

Cytoplasmic and Nuclear Receptors
Estrogen Receptors
Amino Acids
Estrogen Receptor Modulators
Sucrose

Cloning of the rat progesterone receptor gene 5'-region and identification of two functionally distinct promoters

Kraus, W. L., Montano, M. M. & Katzenellenbogen, B. S., Dec 1993, In : Molecular Endocrinology. 7, 12, p. 1603-1616 14 p.

Research output: Contribution to journalArticle

Chloramphenicol O-Acetyltransferase
Progesterone Receptors
Organism Cloning
Estrogen Receptors
Genes

Coactivator peptides have a differential stabilizing effect on the binding of Estrogens and Antiestrogens with the estrogen receptor

Gee, A. C., Carlson, K. E., Martini, P. G. V., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 1 1999, In : Molecular Endocrinology. 13, 11, p. 1912-1923 12 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Nuclear Receptor Coactivator 1
Ligands
Proteolysis
Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Affinity Labels

Comparative effects of estrogen and antiestrogen on plasma renin substrate levels and hepatic estrogen receptors in the rat

Kneifel, M. A. & Katzenellenbogen, B. S., Feb 1981, In : Endocrinology. 108, 2, p. 545-552 8 p.

Research output: Contribution to journalArticle

Angiotensinogen
Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Cytoplasmic and Nuclear Receptors
Estrogen Receptor Modulators
Uterus
Estradiol
Estrogens
Breast Neoplasms

Comprehensive assessment of estrogen receptor beta antibodies in cancer cell line models and tissue reveals critical limitations in reagent specificity

Nelson, A. W., Groen, A. J., Miller, J. L., Warren, A. Y., Holmes, K. A., Tarulli, G. A., Tilley, W. D., Katzenellenbogen, B. S., Hawse, J. R., Gnanapragasam, V. J. & Carroll, J. S., Jan 15 2017, In : Molecular and Cellular Endocrinology. 440, p. 138-150 13 p.

Research output: Contribution to journalArticle

Estrogen Receptor beta
Estrogen Receptors
Cells
Tissue
Cell Line
Estrogen Receptors
Ligands
Estradiol
Estrogens
Aptitude

Considerations in the design and evaluation of cytotoxic estrogens

Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Dec 1 1982, In : Breast Cancer Research and Treatment. 2, 4, p. 347-353 7 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Breast Neoplasms
Estradiol
DNA

Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein

Weis, K. E., Ekena, K., Thomas, J. A., Lazennec, G. & Katzenellenbogen, B. S., Dec 1 1996, In : Molecular Endocrinology. 10, 11, p. 1388-1398 11 p.

Research output: Contribution to journalArticle

Amino Acid Substitution
Estrogen Receptors
Tyrosine
Nuclear Receptor Coactivator 1
Estrogens
Estrogen Receptors
Chromatin
Formaldehyde
Breast Neoplasms
Ligands

Cyclin D1 antagonizes BRCA1 repression of estrogen receptor α activity

Wang, C., Fan, S., Li, Z., Fu, M., Rao, M., Ma, Y., Lisanti, M. P., Albanese, C., Katzenellenbogen, B. S., Kushner, P. J., Weber, B., Rosen, E. M. & Pestell, R. G., Aug 1 2005, In : Cancer Research. 65, 15, p. 6557-6567 11 p.

Research output: Contribution to journalArticle

Cyclin D1
Estrogen Receptors
Response Elements
Estrogens
Breast Neoplasms

Derivation and analysis of a lag-decay model for protein turnover involving a biosynthetic precursor

Katzenellenbogen, J. A., Scheeline, A., Mullick, A. & Katzenellenbogen, B. S., Jan 1 1986, In : Journal of Biological Chemistry. 261, 28, p. 13244-13246 3 p.

Research output: Contribution to journalArticle

Proteins

Design of pathway preferential estrogens that provide beneficial metabolic and vascular effects without stimulating reproductive tissues

Madak-Erdogan, Z., Kim, S. H., Gong, P., Zhao, Y. C., Zhang, H., Chambliss, K. L., Carlson, K. E., Mayne, C. G., Shaul, P. W., Korach, K. S., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., May 24 2016, In : Science Signaling. 9, 429, ra53.

Research output: Contribution to journalArticle

Blood Vessels
Estrogens
Tissue
Ligands
Estrogen Receptors
Progesterone Receptors
Estrogen Receptors
Ligands
Estrogens
Response Elements

Determinants of ligand specificity of estrogen receptor-α: Estrogen versus androgen discrimination

Ekena, K., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 9 1998, In : Journal of Biological Chemistry. 273, 2, p. 693-699 7 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Androgens
Estrogens
Ligands
Estradiol

Dietary licorice root supplementation reduces diet-induced weight gain, lipid deposition, and hepatic steatosis in ovariectomized mice without stimulating reproductive tissues and mammary gland

Madak-Erdogan, Z., Gong, P., Zhao, Y. C., Xu, L., Wrobel, K. U., Hartman, J. A., Wang, M., Cam, A., Iwaniec, U. T., Turner, R. T., Twaddle, N. C., Doerge, D. R., Khan, I. A., Katzenellenbogen, J. A., Katzenellenbogen, B. S. & Helferich, W. G., Feb 1 2016, In : Molecular Nutrition and Food Research. 60, 2, p. 369-380 12 p.

Research output: Contribution to journalArticle

Glycyrrhiza
licorice
fatty liver
Human Mammary Glands
mammary glands
Estrogen Receptor Modulators
Response Elements
Estrogen Receptors
Estradiol
DNA
Keratin-13
Selective Estrogen Receptor Modulators
Gene expression
Estradiol
Estrogen Receptors
Gene Expression Regulation
Estrogen Receptors
Estrogens
Breast Neoplasms
Messenger RNA
Selective Estrogen Receptor Modulators
Conjugated (USP) Estrogens
Cytoplasmic and Nuclear Receptors
Estrogens
Tissue
Estrogen Receptor Modulators
Transcription
Transcriptional Activation
Estradiol
Chemical activation

Different residues of the human estrogen receptor are involved in the recognition of structurally diverse estrogens and antiestrogens

Ekena, K., Weise, K. E., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Feb 21 1997, In : Journal of Biological Chemistry. 272, 8, p. 5069-5075 7 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Ligands
Estradiol

Direct Acetylation of the Estrogen Receptor α Hinge Region by p300 Regulates Transactivation and Hormone Sensitivity

Wang, C., Fu, M., Angeletti, R. H., Siconolfi-Baez, L., Reutens, A. T., Albanese, C., Lisanti, M. P., Katzenellenbogen, B. S., Kato, S., Hopp, T., Fuqua, S. A. W., Lopez, G. N., Kushner, P. J. & Pestell, R. G., Jan 25 2001, In : Journal of Biological Chemistry. 276, 21, p. 18375-18383 9 p.

Research output: Contribution to journalArticle

Acetylation
Hinges
Estrogen Receptors
Transcriptional Activation
Hormones

Directed evolution of human estrogen receptor variants with significantly enhanced androgen specificity and affinity

Chen, Z., Katzenellenbogen, B. S., Katzenellenbogen, J. A. & Zhao, H., Aug 6 2004, In : Journal of Biological Chemistry. 279, 32, p. 33855-33864 10 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Androgens
Ligands
Testosterone
Cytoplasmic and Nuclear Receptors