Benita S Katzenellenbogen

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2001

Nongenotropic, sex-nonspecific signaling through the estrogen or androgen receptors: Dissociation from transcriptional activity

Kousteni, S., Bellido, T., Plotkin, L. I., O'Brien, C. A., Bodenner, D. L., Han, L., Han, K., DiGregorio, G. B., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Roberson, P. K., Weinstein, R. S., Jilka, R. L. & Manolagas, S. C., Mar 9 2001, In : Cell. 104, 5, p. 719-730 12 p.

Research output: Contribution to journalArticle

Open Access

Structure-function relationships in estrogen receptors and the characterization of novel selective estrogen receptor modulators with unique pharmacological profiles

Katzenellenbogen, B. S., Sun, J., Harrington, W. R., Kraichely, D. M., Ganessunker, D. & Katzenellenbogen, J. A., 2001, In : Annals of the New York Academy of Sciences. 949, p. 6-15 10 p.

Research output: Contribution to journalArticle

Synergistic activation of the serotonin-1A receptor by nuclear factor-κB and estrogen

Wissink, S., Van Der Burg, B., Katzenellenbogen, B. S. & Van Der Saag, P. T., 2001, In : Molecular Endocrinology. 15, 4, p. 543-552 10 p.

Research output: Contribution to journalArticle

Synthesis and biological evaluation of a novel series of furans: Ligands selective for estrogen receptor α

Mortensen, D. S., Rodriguez, A. L., Carlson, K. E., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Nov 8 2001, In : Journal of Medicinal Chemistry. 44, 23, p. 3838-3848 11 p.

Research output: Contribution to journalArticle

The estrogen receptor: A structure-based approach to the design of new specific hormone-receptor combinations

Tedesco, R., Thomas, J. A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Apr 25 2001, In : Chemistry and Biology. 8, 3, p. 277-287 11 p.

Research output: Contribution to journalArticle

Triarylpyrazoles with basic side chains: Development of pyrazole-based estrogen receptor antagonists

Stauffer, S. R., Huang, Y. R., Aron, Z. D., Coletta, C. J., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 8 2001, In : Bioorganic and Medicinal Chemistry. 9, 1, p. 151-161 11 p.

Research output: Contribution to journalArticle

2000

Activation of estrogen receptor-α by the heavy metal cadmium

Stoica, A., Katzenellenbogen, B. S. & Martin, M. B., 2000, In : Molecular Endocrinology. 14, 4, p. 545-553 9 p.

Research output: Contribution to journalArticle

Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction

Stauffer, S. R., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jun 1 2000, In : Bioorganic and Medicinal Chemistry. 8, 6, p. 1293-1316 24 p.

Research output: Contribution to journalArticle

Analysis of estrogen receptor interaction with a repressor of estrogen receptor activity (REA) and the regulation of estrogen receptor transcriptional activity by REA

Delage-Mourroux, R., Martini, P. G. V., Choi, I., Kraichely, D. M., Hoeksema, J. & Katzenellenbogen, B. S., Nov 17 2000, In : Journal of Biological Chemistry. 275, 46, p. 35848-35856 9 p.

Research output: Contribution to journalArticle

A role for Akt in mediating the estrogenic functions of epidermal growth factor and insulin-like growth factor I

Martin, M. B., Franke, T. F., Stoica, G. E., Chambon, P., Katzenellenbogen, B. S., Stoica, B. A., McLemore, M. S., Olivo, S. E. & Stoica, A., 2000, In : Endocrinology. 141, 12, p. 4503-4511 9 p.

Research output: Contribution to journalArticle

Estrogen receptor-KRAB chimeras are potent ligand-dependent repressors of estrogen-regulated gene expression

De Haan, G., Chusacultanachai, S., Mao, C., Katzenellenbogen, B. S. & Shapiro, D. J., May 5 2000, In : Journal of Biological Chemistry. 275, 18, p. 13493-13501 9 p.

Research output: Contribution to journalArticle

Estrogen receptors: Selective ligands, partners, and distinctive pharmacology

Katzenellenbogen, B. S., Montano, M. M., Ediger, T. R., Sun, J., Ekena, K., Lazennec, G., Martini, P. G. V., McInerney, E. M., Delage-Mourroux, R., Weis, K., Katzenellenbogen, J. A., Nagel, S., Schrader, W., Bethea, C., Cutler, G. & Hock, J., 2000, In : Recent Progress in Hormone Research. 55, p. 163-195 33 p.

Research output: Contribution to journalArticle

Molecular mechanisms of estrogen action: Selective ligands and receptor pharmacology

Katzenellenbogen, B. S., Choi, I., Delage-Mourroux, R., Ediger, T. R., Martini, P. G. V., Montano, M., Sun, J., Weis, K. & Katzenellenbogen, J. A., Nov 30 2000, In : Journal of Steroid Biochemistry and Molecular Biology. 74, 5, p. 279-285 7 p.

Research output: Contribution to journalArticle

Multistep signaling and transcriptional requirements for pituitary organogenesis in vivo

Rosenfeld, M. G., Briata, P., Dasen, J., Gleiberman, A. S., Kioussi, C., Lin, C., O'Connell, S. M., Ryan, A., Szeto, D. P., Treier, M., Katzenellenbogen, B., Nilson, J., Lawrence, A., Arnhold, I., Frohman, L. & Kochupillai, N., Dec 1 2000, In : Recent Progress in Hormone Research. 55, p. 1-14 14 p.

Research output: Contribution to journalArticle

Prothymosin alpha selectively enhances estrogen receptor transcriptional activity by interacting with a repressor of estrogen receptor activity

Martini, P. G. V., Delage-Mourroux, R., Kraichely, D. M. & Katzenellenbogen, B. S., 2000, In : Molecular and cellular biology. 20, 17, p. 6224-6232 9 p.

Research output: Contribution to journalArticle

Pyrazole ligands: Structure - Affinity/activity relationships and estrogen receptor-α-selective agonists

Stauffer, S. R., Coletta, C. J., Tedesco, R., Nishiguchi, G., Carlson, K., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 28 2000, In : Journal of Medicinal Chemistry. 43, 26, p. 4934-4947 14 p.

Research output: Contribution to journalArticle

1999

Analysis of estrogen response element binding by genetically selected steroid receptor DNA binding domain mutants exhibiting altered specificity and enhanced affinity

Chusacultanachai, S., Glenn, K. A., Rodriguez, A. O., Read, E. K., Gardner, J. F., Katzenellenbogen, B. S. & Shapiro, D. J., Aug 13 1999, In : Journal of Biological Chemistry. 274, 33, p. 23591-23598 8 p.

Research output: Contribution to journalArticle

An estrogen receptor-selective coregulator that potentiates the effectiveness of antiestrogens and represses the activity of estrogens

Montano, M. M., Ekena, K., Delage-Mourroux, R., Chang, W., Martini, P. & Katzenellenbogen, B. S., Jun 8 1999, In : Proceedings of the National Academy of Sciences of the United States of America. 96, 12, p. 6947-6952 6 p.

Research output: Contribution to journalArticle

Caveolin-1 potentiates estrogen receptor α (ERα) signaling. Caveolin-1 drives ligand-independent nuclear translocation and activation of ERα

Schlegel, A., Wang, C., Katzenellenbogen, B. S., Pestell, R. G. & Lisanti, M. P., Nov 19 1999, In : Journal of Biological Chemistry. 274, 47, p. 33551-33556 6 p.

Research output: Contribution to journalArticle

Coactivator peptides have a differential stabilizing effect on the binding of Estrogens and Antiestrogens with the estrogen receptor

Gee, A. C., Carlson, K. E., Martini, P. G. V., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., 1999, In : Molecular Endocrinology. 13, 11, p. 1912-1923 12 p.

Research output: Contribution to journalArticle

Estrogen receptor regulation of the Na+/H+ exchanger regulatory factor

Ediger, T. R., Kraus, W. L., Weinman, E. J. & Katzenellenbogen, B. S., 1999, In : Endocrinology. 140, 7, p. 2976-2982 7 p.

Research output: Contribution to journalArticle

Estrogen receptor subtype-selective ligands: Asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl-5,6,11,12- tetrahydrochrysenes

Meyers, M. J., Jun, S., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jul 1 1999, In : Journal of Medicinal Chemistry. 42, 13, p. 2456-2468 13 p.

Research output: Contribution to journalArticle

Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-α or estrogen receptor-β

Sun, J., Meyers, M. J., Fink, B. E., Rajendran, R., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., 1999, In : Endocrinology. 140, 2, p. 800-804 5 p.

Research output: Contribution to journalArticle

The estrogen receptor enhances AP-1 activity by two distinct mechanisms with different requirements for receptor transactivation functions

Webb, P., Nguyen, P., Valentine, C., Lopez, G. N., Kwok, G. R., McInerney, E., Katzenellenbogen, B. S., Enmark, E., Gustafsson, J. Å., Nilsson, S. & Kushner, P. J., 1999, In : Molecular Endocrinology. 13, 10, p. 1672-1685 14 p.

Research output: Contribution to journalArticle

1998

Determinants of ligand specificity of estrogen receptor-α: Estrogen versus androgen discrimination

Ekena, K., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 9 1998, In : Journal of Biological Chemistry. 273, 2, p. 693-699 7 p.

Research output: Contribution to journalArticle

Estrogen receptor activation function 1 works by binding p160 coactivator proteins

Webb, P., Nguyen, P., Shinsako, J., Anderson, C., Feng, W., Nguyen, M. P., Chen, D., Huang, S. M., Subramanian, S., McKinerney, E., Katzenellenbogen, B. S., Stallcup, M. R. & Kushner, P. J., 1998, In : Molecular Endocrinology. 12, 10, p. 1605-1618 14 p.

Research output: Contribution to journalArticle

Open Access

Transcription activation by the human estrogen receptor subtype β (ERβ) studied with ERβ and ERα receptor chimeras

Mcinerney, E. M., Weis, K. E., Sun, J., Mosselman, S. & Katzenellenbogen, B. S., 1998, In : Endocrinology. 139, 11, p. 4513-4522 10 p.

Research output: Contribution to journalArticle

Transcriptional regulation of the human quinone reductase gene by antiestrogen-liganded estrogen receptor-α and estrogen receptor-β

Montano, M. M., Jaiswal, A. K. & Katzenellenbogen, B. S., Sep 25 1998, In : Journal of Biological Chemistry. 273, 39, p. 25443-25449 7 p.

Research output: Contribution to journalArticle

1997

17α-(Haloacetamidoalkyl)estradiols alkylate the human estrogen receptor at cysteine residues 417 and 530

Aliau, S., El Garrouj, D., Yasri, A., Katzenellenbogen, B. S. & Borgna, J. L., May 13 1997, In : Biochemistry. 36, 19, p. 58615867 58615867 p.

Research output: Contribution to journalArticle

Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open pocket conformation is required for ligand interaction

Carlson, K. E., Choi, I., Gee, A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 2 1997, In : Biochemistry. 36, 48, p. 14897-14905 9 p.

Research output: Contribution to journalArticle

Different residues of the human estrogen receptor are involved in the recognition of structurally diverse estrogens and antiestrogens

Ekena, K., Weise, K. E., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Feb 21 1997, In : Journal of Biological Chemistry. 272, 8, p. 5069-5075 7 p.

Research output: Contribution to journalArticle

1996

Analysis of estrogen receptor transcriptional enhancement by a nuclear hormone receptor coactivator

Mcinerney, E. M., Tsai, M. J., O'Malley, B. W. & Katzenellenbogen, B. S., Sep 17 1996, In : Proceedings of the National Academy of Sciences of the United States of America. 93, 19, p. 10069-10073 5 p.

Research output: Contribution to journalArticle

A transcriptionally active estrogen receptor mutant is a novel type of dominant negative inhibitor of estrogen action

McInerney, E. M., Ince, B. A., Shapiro, D. J. & Katzenellenbogen, B. S., 1996, In : Molecular Endocrinology. 10, 12, p. 1519-1526 8 p.

Research output: Contribution to journalArticle

Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein

Weis, K. E., Ekena, K., Thomas, J. A., Lazennec, G. & Katzenellenbogen, B. S., 1996, In : Molecular Endocrinology. 10, 11, p. 1388-1398 11 p.

Research output: Contribution to journalArticle

Estrogen receptors: Bioactivities and interactions with cell signaling pathways

Katzenellenbogen, B. S., Feb 1996, In : Biology of reproduction. 54, 2, p. 287-293 7 p.

Research output: Contribution to journalArticle

Identification of amino acids in the hormone binding domain of the human estrogen receptor important in estrogen binding

Ekena, K., Weis, K. E., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., 1996, In : Journal of Biological Chemistry. 271, 33, p. 20053-20059 7 p.

Research output: Contribution to journalArticle