Benita S Katzenellenbogen

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Research Output

Article

Antagonists for Constitutively Active Mutant Estrogen Receptors: Insights into the Roles of Antiestrogen-Core and Side-Chain

Sharma, A., Toy, W., Guillen, V. S., Sharma, N., Min, J., Carlson, K. E., Mayne, C. G., Lin, S., Sabio, M., Greene, G., Katzenellenbogen, B. S., Chandarlapaty, S. & Katzenellenbogen, J. A., Dec 21 2018, In : ACS chemical biology. 13, 12, p. 3374-3384 11 p.

Research output: Contribution to journalArticle

Antagonists selective for estrogen receptor α

Sun, J., Huang, Y. R., Harrington, W. R., Sheng, S., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., 2002, In : Endocrinology. 143, 3, p. 941-947 7 p.

Research output: Contribution to journalArticle

Antiestrogen action in the uterus: Biological ineffectiveness of nuclear bound estradiol after antiestrogen

Katzenellenbogen, B. S. & Ferguson, E. R., Jun 1975, In : Endocrinology. 97, 1, p. 1-12 12 p.

Research output: Contribution to journalArticle

Antiestrogen Binding in Antiestrogen Growth-resistant Estrogen-responsive Clonal Variants of MCF-7 Human Breast Cancer Cells

Miller, M. A., Lippman, M. E. & Katzenellenbogen, B. S., Nov 1 1984, In : Cancer Research. 44, 11, p. 5038-5045 8 p.

Research output: Contribution to journalArticle

Antiestrogenic Potency and Binding Characteristics of the Triphenylethylene H1285 in MCF-7 Human Breast Cancer Cells

Sheen, Y. Y., Ruh, T. S., Mangel, W. F. & Katzenellenbogen, B. S., Sep 1 1985, In : Cancer Research. 45, 9, p. 4192-4199 8 p.

Research output: Contribution to journalArticle

Anti-estrogen interaction with uterine estrogen receptors. Studies with a radiolabeled anti-estrogen (CI-628)

Katzenellenbogen, B. S., Katzenellenbogen, J. A., Ferguson, E. R. & Krauthammer, N., Dec 1 1978, In : Journal of Biological Chemistry. 253, 3, p. 697-707 11 p.

Research output: Contribution to journalArticle

Antiestrogen Modulation of the Growth and Properties of Ovarian-Autonomous and Ovarian-Dependent Mammary Tumors in Rats

Tsai, T. L. S., Rutledge, S. & Katzenellenbogen, B. S., Dec 1 1979, In : Cancer Research. 39, 12, p. 5043-5050 8 p.

Research output: Contribution to journalArticle

Antiestrogen pharmacology and mechanism of action

Katzenellenbogen, B. S., Miller, M. A., Eckert, R. L. & Sudo, K., 1983, In : Journal of Steroid Biochemistry. 19, 1, p. 59-68 10 p.

Research output: Contribution to journalArticle

Antiestrogens: Studies using an in vitro estrogen-responsive uterine system

Katzenellebogen, B. S. & Katzenellenbogen, J. A., Feb 20 1973, In : Biochemical and Biophysical Research Communications. 50, 4, p. 1152-1159 8 p.

Research output: Contribution to journalArticle

Antiestrogens: Mechanisms and actions in target cells

Katzenellenbogen, B. S., Montano, M. M., Le Goff, P., Schodin, D. J., Kraus, W. L., Bhardwaj, B. & Fujimoto, N., Jun 1995, In : Journal of Steroid Biochemistry and Molecular Biology. 53, 1-6, p. 387-393 7 p.

Research output: Contribution to journalArticle

A repressive role for prohibitin in estrogen signaling

He, B., Feng, Q., Mukherjee, A., Lonard, D. M., DeMayo, F. J., Katzenellenbogen, B. S., Lydon, J. P. & O'Malley, B. W., Feb 2008, In : Molecular Endocrinology. 22, 2, p. 344-360 17 p.

Research output: Contribution to journalArticle

A role for Akt in mediating the estrogenic functions of epidermal growth factor and insulin-like growth factor I

Martin, M. B., Franke, T. F., Stoica, G. E., Chambon, P., Katzenellenbogen, B. S., Stoica, B. A., McLemore, M. S., Olivo, S. E. & Stoica, A., 2000, In : Endocrinology. 141, 12, p. 4503-4511 9 p.

Research output: Contribution to journalArticle

A transcriptionally active estrogen receptor mutant is a novel type of dominant negative inhibitor of estrogen action

McInerney, E. M., Ince, B. A., Shapiro, D. J. & Katzenellenbogen, B. S., 1996, In : Molecular Endocrinology. 10, 12, p. 1519-1526 8 p.

Research output: Contribution to journalArticle

Bibenzyl- and stilbene-core compounds with non-polar linker atom substituents as selective ligands for estrogen receptor beta

Waibel, M., De Angelis, M., Stossi, F., Kieser, K. J., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Sep 2009, In : European Journal of Medicinal Chemistry. 44, 9, p. 3412-3424 13 p.

Research output: Contribution to journalArticle

Bioactivities, Estrogen Receptor Interactions, and Plasminogen Activator-inducing Activities of Tamoxifen and Hydroxy-tamoxifen Isomers in MCF-7 Human Breast Cancer Cells

Katzenellenbogen, B. S., Norman, M. J., Eckert, R. L., Peltz, S. W. & Mangel, W. F., Jan 1 1984, In : Cancer Research. 44, 1, p. 112-119 8 p.

Research output: Contribution to journalArticle

Biological activities of tamoxifen aziridine, an antiestrogen-based affinity label for the estrogen receptor, in vivo and in vitro

Wei, L. L., Mangel, W. F. & Katzenellenbogen, B. S., Dec 1985, In : Journal of Steroid Biochemistry. 23, 6 PART 1, p. 875-881 7 p.

Research output: Contribution to journalArticle

Biological Activity and Receptor Binding of a Strongly Interacting Estrogen in Human Breast Cancer Cells

Reiner, G. C. A., Katzenellenbogen, B. S., Bindal, R. D. & Katzenellenbogen, J. A., Jun 1 1984, In : Cancer Research. 44, 6, p. 2302-2308 7 p.

Research output: Contribution to journalArticle

Biological Potency and Uterine Estrogen Receptor Interactions of the Metabolites of the Antiestrogens CI628 and U23, 469

Hayes, J. R., Rorke, E. A., Robertson, D. W., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 1981, In : Endocrinology. 108, 1, p. 164-172 9 p.

Research output: Contribution to journalArticle

Biology and receptor interactions of estriol and estriol derivatives in vitro and in vivo

Katzenellenbogen, B. S., Apr 1984, In : Journal of Steroid Biochemistry. 20, 4 PART 2, p. 1033-1037 5 p.

Research output: Contribution to journalArticle

Bivalent ligands as probes of estrogen receptor action

Bergmann, K. E., Wooge, C. H., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jun 1994, In : Journal of Steroid Biochemistry and Molecular Biology. 49, 2-3, p. 139-152 14 p.

Research output: Contribution to journalArticle

Bridged bicyclic cores containing a 1,1-diarylethylene motif are high-affinity subtype-selective ligands for the estrogen receptor

Muthyala, R. S., Sheng, S., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Apr 24 2003, In : Journal of Medicinal Chemistry. 46, 9, p. 1589-1602 14 p.

Research output: Contribution to journalArticle

Caveolin-1 potentiates estrogen receptor α (ERα) signaling. Caveolin-1 drives ligand-independent nuclear translocation and activation of ERα

Schlegel, A., Wang, C., Katzenellenbogen, B. S., Pestell, R. G. & Lisanti, M. P., Nov 19 1999, In : Journal of Biological Chemistry. 274, 47, p. 33551-33556 6 p.

Research output: Contribution to journalArticle

Characterization and regulation of estrogen and progesterone receptors in breast cancer.

Read, L. D. & Katzenellenbogen, B. S., Dec 1 1992, In : Cancer treatment and research. 61, p. 277-299 23 p.

Research output: Contribution to journalArticle

Characterization of the biological roles of the estrogen receptors, ERα and ERβ, in estrogen target tissues in vivo through the use of an ERα-selective ligand

Harris, H. A., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Nov 1 2002, In : Endocrinology. 143, 11, p. 4172-4177 6 p.

Research output: Contribution to journalArticle

Characterization of the estrogen receptor and its dynamics in MCF-7 human breast cancer cells using a covalently attaching antiestrogen

Monsma, F. J., Katzenellenbogen, B. S., Miller, M. A., Ziegler, Y. S. & Katzenellenbogen, J. A., 1984, In : Endocrinology. 115, 1, p. 143-153 11 p.

Research output: Contribution to journalArticle

Characterization of the interactions of estrogen receptor and MNAR in the activation of cSrc

Barletta, F., Wong, C. W., McNally, C., Komm, B. S., Katzenellenbogen, B. & Cheskis, B. J., May 2004, In : Molecular Endocrinology. 18, 5, p. 1096-1108 13 p.

Research output: Contribution to journalArticle

Characterization of the pharmacophore properties of novel selective estrogen receptor downregulators (SERDs)

Kieser, K. J., Kim, D. W., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Apr 22 2010, In : Journal of Medicinal Chemistry. 53, 8, p. 3320-3329 10 p.

Research output: Contribution to journalArticle

Characterization of the subunit nature of nuclear estrogen receptors by chemical cross-linking and dense amino acid labeling

Miller, M. A., Mullick, A., Greene, G. L. & Katzenellenbogen, B. S., Aug 1985, In : Endocrinology. 117, 2, p. 515-522 8 p.

Research output: Contribution to journalArticle

Cloning of the rat progesterone receptor gene 5'-region and identification of two functionally distinct promoters

Kraus, W. L., Montano, M. M. & Katzenellenbogen, B. S., Dec 1993, In : Molecular Endocrinology. 7, 12, p. 1603-1616 14 p.

Research output: Contribution to journalArticle

Coactivator peptides have a differential stabilizing effect on the binding of Estrogens and Antiestrogens with the estrogen receptor

Gee, A. C., Carlson, K. E., Martini, P. G. V., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., 1999, In : Molecular Endocrinology. 13, 11, p. 1912-1923 12 p.

Research output: Contribution to journalArticle

Combined Targeting of Estrogen Receptor Alpha and Exportin 1 in Metastatic Breast Cancers

Cotul, E. K., Zuo, Q., Santaliz-Casiano, A., Imir, O. B., Mogol, A. N., Tunc, E., Duong, K., Lee, J. K., Ramesh, R., Odukoya, E., Kesavadas, M. P., Ziogaite, M., Smith, B. P., Mao, C., Shapiro, D. J., Park, B. H., Katzenellenbogen, B. S., Daly, D., Aranda, E., O’Neill, J. D. & 3 others, Walker, C., Landesman, Y. & Madak-Erdogan, Z., Aug 22 2020, In : Cancers. 12, 9, 2397.

Research output: Contribution to journalArticle

Open Access

Comparative effects of estrogen and antiestrogen on plasma renin substrate levels and hepatic estrogen receptors in the rat

Kneifel, M. A. & Katzenellenbogen, B. S., Feb 1981, In : Endocrinology. 108, 2, p. 545-552 8 p.

Research output: Contribution to journalArticle

Comprehensive assessment of estrogen receptor beta antibodies in cancer cell line models and tissue reveals critical limitations in reagent specificity

Nelson, A. W., Groen, A. J., Miller, J. L., Warren, A. Y., Holmes, K. A., Tarulli, G. A., Tilley, W. D., Katzenellenbogen, B. S., Hawse, J. R., Gnanapragasam, V. J. & Carroll, J. S., Jan 15 2017, In : Molecular and Cellular Endocrinology. 440, p. 138-150 13 p.

Research output: Contribution to journalArticle

Considerations in the design and evaluation of cytotoxic estrogens

Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Dec 1 1982, In : Breast Cancer Research and Treatment. 2, 4, p. 347-353 7 p.

Research output: Contribution to journalArticle

Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein

Weis, K. E., Ekena, K., Thomas, J. A., Lazennec, G. & Katzenellenbogen, B. S., 1996, In : Molecular Endocrinology. 10, 11, p. 1388-1398 11 p.

Research output: Contribution to journalArticle