Benita S Katzenellenbogen

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Research Output

Identification of cysteine 530 as the covalent attachment site of an affinity-labeling estrogen (ketononestrol aziridine) and antiestrogen (tamoxifen aziridine) in the human estrogen receptor

Harlow, K. W., Smith, D. N., Katzenellenbogen, J. A., Greene, G. L. & Katzenellenbogen, B. S., 1989, In : Journal of Biological Chemistry. 264, 29, p. 17476-17485 10 p.

Research output: Contribution to journalArticle

Identification of multiple, widely spaced estrogen-responsive regions in the rat progesterone receptor gene

Kraus, W. L., Montano, M. M. & Katzenellenbogen, B. S., Aug 1 1994, In : Molecular Endocrinology. 8, 8, p. 952-969 18 p.

Research output: Contribution to journalArticle

Impact of estrogen receptor β on gene networks regulated by estrogen receptor α in breast cancer cells

Chang, E. C., Frasor, J., Komm, B. & Katzenellenbogen, B. S., Sep 22 2006, In : Endocrinology. 147, 10, p. 4831-4842 12 p.

Research output: Contribution to journalArticle

Inactive proteinases in silkmoth moulting gel

Katzenellenbogen, B. S. & Kafatos, F. C., May 1971, In : Journal of insect physiology. 17, 5, p. 823-832 10 p.

Research output: Contribution to journalArticle

Indazole estrogens: Highly selective ligands for the estrogen receptor β

De Angelis, M., Stossi, F., Carlson, K. A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Feb 24 2005, In : Journal of Medicinal Chemistry. 48, 4, p. 1132-1144 13 p.

Research output: Contribution to journalArticle

In memoriam: Jack Gorski (1931-2006).

Katzenellenbogen, B. S., Nov 2006, In : Molecular endocrinology (Baltimore, Md.). 20, 11, p. 2611-2612 2 p.

Research output: Contribution to journalArticle

Integrative genomics of gene and metabolic regulation by estrogen receptors α and β, and their coregulators

Madak-Erdogan, Z., Charn, T. H., Jiang, Y., Liu, E. T., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 2013, In : Molecular Systems Biology. 9, 201328.

Research output: Contribution to journalArticle

Interaction of a high affinity anti-estrogen (α-[4-pyrrolidinoethoxy]phenyl-4-hydroxy-α'-nitrostilbene, CI628M) with uterine estrogen receptors

Katzenellenbogen, B. S., Pavlik, E. J., Robertson, D. W. & Katzenellenbogen, J. A., Jan 1 1981, In : Journal of Biological Chemistry. 256, 6, p. 2908-2915 8 p.

Research output: Contribution to journalArticle

Iodohexestrols. II. Characterization of the Binding and Estrogenic Activity of Iodinated Hexestrol Derivatives, in Vitro and in Vivo

Katzenellenbogen, J. A., Hsiung, H. M., Carlson, K. E., Mcguire, W. L., Kraay, R. J. & Katzenellenbogen, B. S., Apr 1 1975, In : Biochemistry. 14, 8, p. 1742-1750 9 p.

Research output: Contribution to journalArticle

Isocoumarins as estrogen receptor beta selective ligands: Isomers of isoflavone phytoestrogens and their metabolites

De Angelis, M., Stossi, F., Waibel, M., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 1 2005, In : Bioorganic and Medicinal Chemistry. 13, 23, p. 6529-6542 14 p.

Research output: Contribution to journalArticle

Ketononestrol aziridine, an agonistic estrogen receptor affinity label: Study of its bioactivity and estrogen receptor covalent labeling

Elliston, J. F., Zablocki, J. A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Aug 1 1987, In : Endocrinology. 121, 2, p. 667-676 10 p.

Research output: Contribution to journalArticle

Licorice root components in dietary supplements are selective estrogen receptor modulators with a spectrum of estrogenic and anti-estrogenic activities

Boonmuen, N., Gong, P., Ali, Z., Chittiboyina, A. G., Khan, I., Doerge, D. R., Helferich, W. G., Carlson, K. E., Martin, T., Piyachaturawat, P., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 2016, In : Steroids. 105, p. 42-49 8 p.

Research output: Contribution to journalArticle

Ligand accessibility and bioactivity of a hormone-dendrimer conjugate depend on pH and pH history

Kim, S. H., Madak-Erdogan, Z., Bae, S. C., Carlson, K. E., Mayne, C. G., Granick, S., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Aug 19 2015, In : Journal of the American Chemical Society. 137, 32, p. 10326-10335 10 p.

Research output: Contribution to journalArticle

Ligand-modulated regulation of progesterone receptor messenger ribonucleic acid and protein in human breast cancer cell lines

Read, L. D., Snider, C. E., Miller, J. S., Greene, G. L. & Katzenellenbogen, B. S., Mar 1988, In : Molecular Endocrinology. 2, 3, p. 263-271 9 p.

Research output: Contribution to journalArticle

Lipin1 regulation by estrogen in uterus and liver: Implications for diabetes and fertility

Gowri, P. M., Sengupta, S., Bertera, S. & Katzenellenbogen, B. S., Aug 1 2007, In : Endocrinology. 148, 8, p. 3685-3693 9 p.

Research output: Contribution to journalArticle

Lipophilic impurities, not phenolsulfonphthalein, account for the estrogenic activity in commercial preparations of phenol red

Bindal, R. D., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Sep 1988, In : Journal of Steroid Biochemistry. 31, 3, p. 287-293 7 p.

Research output: Contribution to journalArticle

Localization of androgen and estrogen receptors in adult male mouse reproductive tract

Zhou, Q., Nie, R., Prins, G. S., Saunders, P. T. K., Katzenellenbogen, B. S. & Hess, R. A., Nov 1 2002, In : Journal of andrology. 23, 6, p. 870-881 12 p.

Research output: Contribution to journalArticle

Localization of estrogen receptors in uterine cells. An appraisal of translocation

Pavlik, E. J., Rutledge, S., Eckert, R. L. & Katzenellenbogen, B. S., Oct 1 1979, In : Experimental Cell Research. 123, 1, p. 177-189 13 p.

Research output: Contribution to journalArticle

Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens

Jiang, Y., Gong, P., Madak-Erdogan, Z., Martin, T., Jeyakumar, M., Carlson, K., Khan, I., Smillie, T. J., Chittiboyina, A. G., Rotte, S. C. K., Helferich, W. G., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Nov 1 2013, In : FASEB Journal. 27, 11, p. 4406-4418 13 p.

Research output: Contribution to journalArticle

Mechanisms of estrogen and antiestrogen action in mammary cancer

Katzenellenbogen, B. S., Rorke, E. A. & Eckert, R. L., Dec 1981, In : Journal of Steroid Biochemistry. 15, C, p. 219-229 11 p.

Research output: Contribution to journalArticle

Membrane and nuclear estrogen receptor alpha actions: From tissue specificity to medical implications

Arnal, J. F., Lenfant, F., Metivier, R., Flouriot, G., Henrion, D., Adlanmerini, M., Fontaine, C., Gourdy, P., Chambon, P., Katzenellenbogen, B. & Katzenellenbogen, J., Jul 2017, In : Physiological Reviews. 97, 3, p. 1045-1087 43 p.

Research output: Contribution to journalReview article

Metabolite ligands of estrogen receptor-β reduce primate coronary hyperreactivity

Mishra, R. G., Stanczyk, F. Z., Burry, K. A., Oparil, S., Katzenellenbogen, B. S., Nealen, M. L., Katzenellenbogen, J. A. & Hermsmeyer, R. K., Jan 1 2006, In : American Journal of Physiology - Heart and Circulatory Physiology. 290, 1, p. H295-H303

Research output: Contribution to journalArticle

MMTV-PyMT and Derived Met-1 Mouse Mammary Tumor Cells as Models for Studying the Role of the Androgen Receptor in Triple-Negative Breast Cancer Progression

Christenson, J. L., Butterfield, K. T., Spoelstra, N. S., Norris, J. D., Josan, J. S., Pollock, J. A., McDonnell, D. P., Katzenellenbogen, B. S., Katzenellenbogen, J. A. & Richer, J. K., Apr 1 2017, In : Hormones and Cancer. 8, 2, p. 69-77 9 p.

Research output: Contribution to journalArticle

Modulation of estrogen receptor activity by selective coregulators

Martini, P. G. V. & Katzenellenbogen, B. S., Jun 2003, In : Journal of Steroid Biochemistry and Molecular Biology. 85, 2-5, p. 117-122 6 p.

Research output: Contribution to journalArticle

Molecular basis for the subtype discrimination of the estrogen receptor-β-selective ligand, diarylpropionitrile

Sun, J., Baudry, J., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Feb 1 2003, In : Molecular Endocrinology. 17, 2, p. 247-258 12 p.

Research output: Contribution to journalArticle

Molecular cloning of porcine estrogen receptor-β complementary DNAs and developmental expression in periimplantation embryos

Kowalski, A. A., Graddy, L. G., Vale-Cruz, D. S., Choi, I., Katzenellenbogen, B. S., Simmen, F. A. & Simmen, R. C. M., Jan 1 2002, In : Biology of reproduction. 66, 3, p. 760-769 10 p.

Research output: Contribution to journalArticle

Molecular mechanisms of estrogen action: Selective ligands and receptor pharmacology

Katzenellenbogen, B. S., Choi, I., Delage-Mourroux, R., Ediger, T. R., Martini, P. G. V., Montano, M., Sun, J., Weis, K. & Katzenellenbogen, J. A., Nov 30 2000, In : Journal of Steroid Biochemistry and Molecular Biology. 74, 5, p. 279-285 7 p.

Research output: Contribution to journalArticle

Monoaryl-substituted salicylaldoximes as ligands for estrogen receptor β

Minutolo, F., Bellini, R., Bertini, S., Carboni, I., Lapucci, A., Pistolesi, L., Prota, G., Rapposelli, S., Solati, F., Tuccinardi, T., Martinelli, A., Stossi, F., Carlson, K. E., Katzenellenbogen, B. S., Katzenellenbogen, J. A. & Macchia, M., Mar 13 2008, In : Journal of Medicinal Chemistry. 51, 5, p. 1344-1351 8 p.

Research output: Contribution to journalArticle

Multiple beneficial roles of repressor of estrogen receptor activity (REA) in suppressing the progression of endometriosis

Zhao, Y., Chen, Y., Kuang, Y., Bagchi, M. K., Taylor, R. N., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Feb 2016, In : Endocrinology. 157, 2, p. 900-912 13 p.

Research output: Contribution to journalArticle

Multistep signaling and transcriptional requirements for pituitary organogenesis in vivo

Rosenfeld, M. G., Briata, P., Dasen, J., Gleiberman, A. S., Kioussi, C., Lin, C., O'Connell, S. M., Ryan, A., Szeto, D. P., Treier, M., Katzenellenbogen, B., Nilson, J., Lawrence, A., Arnhold, I., Frohman, L. & Kochupillai, N., Dec 1 2000, In : Recent Progress in Hormone Research. 55, p. 1-14 14 p.

Research output: Contribution to journalArticle

New Class of Selective Estrogen Receptor Degraders (SERDs): Expanding the Toolbox of PROTAC Degrons

Wang, L., Guillen, V. S., Sharma, N., Flessa, K., Min, J., Carlson, K. E., Toy, W., Braqi, S., Katzenellenbogen, B. S., Katzenellenbogen, J. A., Chandarlapaty, S. & Sharma, A., Aug 9 2018, In : ACS Medicinal Chemistry Letters. 9, 8, p. 803-808 6 p.

Research output: Contribution to journalArticle

NFκB selectivity of estrogen receptor ligands revealed by comparative crystallographic analyses

Nettles, K. W., Bruning, J. B., Gil, G., Nowak, J., Sharma, S. K., Hahm, J. B., Kulp, K., Hochberg, R. B., Zhou, H., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Kim, Y., Joachmiak, A. & Greene, G. L., Apr 2008, In : Nature chemical biology. 4, 4, p. 241-247 7 p.

Research output: Contribution to journalArticle

Nitrosourea and nitrosocarbamate derivatives of the antiestrogen tamoxifen as potential estrogen receptor-mediated cytotoxic agents in human breast cancer cells

Wei, L. L., Katzenellenbogen, B. S., Robertson, D. W., Simpson, D. M. & Katzenellenbogen, J. A., Jun 1 1986, In : Breast Cancer Research and Treatment. 7, 2, p. 77-90 14 p.

Research output: Contribution to journalArticle

Non-estrogenic Xanthohumol Derivatives Mitigate Insulin Resistance and Cognitive Impairment in High-Fat Diet-induced Obese Mice

Miranda, C. L., Johnson, L. A., De Montgolfier, O., Elias, V. D., Ullrich, L. S., Hay, J. J., Paraiso, I. L., Choi, J., Reed, R. L., Revel, J. S., Kioussi, C., Bobe, G., Iwaniec, U. T., Turner, R. T., Katzenellenbogen, B. S., Katzenellenbogen, J. A., Blakemore, P. R., Gombart, A. F., Maier, C. S., Raber, J. & 1 others, Stevens, J. F., Dec 1 2018, In : Scientific reports. 8, 1, 613.

Research output: Contribution to journalArticle

Nongenotropic, sex-nonspecific signaling through the estrogen or androgen receptors: Dissociation from transcriptional activity

Kousteni, S., Bellido, T., Plotkin, L. I., O'Brien, C. A., Bodenner, D. L., Han, L., Han, K., DiGregorio, G. B., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Roberson, P. K., Weinstein, R. S., Jilka, R. L. & Manolagas, S. C., Mar 9 2001, In : Cell. 104, 5, p. 719-730 12 p.

Research output: Contribution to journalArticle

Open Access

Nonnuclear estrogen receptor activation improves hepatic steatosis in female mice

Chambliss, K. L., Barrera, J., Umetani, M., Umetani, J., Kim, S. H., Madak-Erdogan, Z., Huang, L., Katzenellenbogen, B. S., Katzenellenbogen, J. A., Mineo, C. & Shaul, P. W., Jan 1 2016, In : Endocrinology. 157, 10, p. 3731-3741 11 p.

Research output: Contribution to journalArticle

Non-nuclear estrogen receptor alpha activation in endothelium reduces cardiac ischemia-reperfusion injury in mice

Menazza, S., Sun, J., Appachi, S., Chambliss, K. L., Kim, S. H., Aponte, A., Khan, S., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Shaul, P. W. & Murphy, E., Jun 1 2017, In : Journal of Molecular and Cellular Cardiology. 107, p. 41-51 11 p.

Research output: Contribution to journalArticle