Benita S Katzenellenbogen

1970 …2018
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Research Output 1970 2018

[125I]Iododesethyl tamoxifen aziridine: Synthesis and covalent labeling of the estrogen receptor with an iodine-labeled affinity label

Salituro, F. G., Carlson, K. E., Elliston, J. F., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 1 1986, In : Steroids. 48, 5-6, p. 287-313 27 p.

Research output: Contribution to journalArticle

Affinity Labels
Iodine
Estrogen Receptors
Labeling
Competitive Binding

[38] Methods for Assessing Estrogen Effects on New Uterine Protein Synthesis In Vitro

Katzenellenbogen, B. S. & Gorski, J., Jan 1 1975, In : Methods in enzymology. 36, C, p. 444-455 12 p.

Research output: Contribution to journalArticle

Estrogens
Proteins
Tissue
RNA
Rats

14-3-3ζ as a predictor of early time to recurrence and distant metastasis in hormone receptor-positive and -negative breast cancers

Bergamaschi, A., Frasor, J., Borgen, K., Stanculescu, A., Johnson, P., Rowland, K. M., Wiley, E. L. & Katzenellenbogen, B. S., Feb 1 2013, In : Breast Cancer Research and Treatment. 137, 3, p. 689-696 8 p.

Research output: Contribution to journalArticle

Hormones
Breast Neoplasms
Neoplasm Metastasis
Recurrence
Estrogen Receptors

17α-(Haloacetamidoalkyl)estradiols alkylate the human estrogen receptor at cysteine residues 417 and 530

Aliau, S., El Garrouj, D., Yasri, A., Katzenellenbogen, B. S. & Borgna, J. L., May 13 1997, In : Biochemistry. 36, 19, p. 58615867 1 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Cysteine
Estradiol
Hormones
Labeling

A case of premature thelarche with no central cause or genetic variants within the estrogen receptor signaling pathway

Hartmaier, R. J., Walenkamp, M. J. E., Richter, A. S., Wang, J., Katzenellenbogen, B. S., Oesterreich, S. & Wit, J. M., 2009, In : Journal of Pediatric Endocrinology and Metabolism. 22, 8, p. 751-758 8 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Hormones
Breast
Serum

A comparative study of antiestrogen action: temporal patterns of antagonism of estrogen stimulated uterine growth and effects on estrogen receptor levels

Ferguson, E. R., Katzenellenbogen, B. S. & Ferguson, E. R., May 1977, In : Endocrinology. 100, 5, p. 1242-1251 10 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Cytoplasmic and Nuclear Receptors
Estrogen Receptors
Nitromifene
Estrogens

Activation of ERα is necessary for estradiol's anorexigenic effect in female rats

Santollo, J., Katzenellenbogen, B. S., Katzenellenbogen, J. A. & Eckel, L. A., Nov 1 2010, In : Hormones and Behavior. 58, 5, p. 872-877 6 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estradiol
Eating
Hormones

Activation of estrogen receptor-α by the heavy metal cadmium

Stoica, A., Katzenellenbogen, B. S. & Martin, M. B., Dec 1 2000, In : Molecular Endocrinology. 14, 4, p. 545-553 9 p.

Research output: Contribution to journalArticle

Heavy Metals
Cadmium
Estrogen Receptors
Hormones
Estradiol

Activation of estrogen receptor β is a prerequisite for estrogen-dependent upregulation of nitric oxide synthases in neonatal rat cardiac myocytes

Nuedling, S., Karas, R. H., Mendelsohn, M. E., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Meyer, R., Vetter, H. & Grohé, C., Aug 3 2001, In : FEBS Letters. 502, 3, p. 103-108 6 p.

Research output: Contribution to journalArticle

Nitric Oxide Synthase Type II
Cardiac Myocytes
Nitric Oxide Synthase
Estrogen Receptors
Rats
Estrogen Receptor Modulators
Estrogen Receptors
Adenosine
Ligands
1-Methyl-3-isobutylxanthine

Activities of estrogen receptor alpha- and beta-selective ligands at diverse estrogen responsive gene sites mediating transactivation or transrepression

Harrington, W. R., Sheng, S., Barnett, D. H., Petz, L. N., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Aug 29 2003, In : Molecular and Cellular Endocrinology. 206, 1-2, p. 13-22 10 p.

Research output: Contribution to journalArticle

Estrogen Receptor beta
Estrogen Receptor alpha
Transcriptional Activation
Estrogens
Genes

Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction

Stauffer, S. R., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jun 1 2000, In : Bioorganic and Medicinal Chemistry. 8, 6, p. 1293-1316 24 p.

Research output: Contribution to journalArticle

Amides
Estrogen Receptors
Ligands
Benzamides
Acetamides

Adamantyl Antiestrogens with Novel Side Chains Reveal a Spectrum of Activities in Suppressing Estrogen Receptor Mediated Activities in Breast Cancer Cells

Min, J., Guillen, V. S., Sharma, A., Zhao, Y., Ziegler, Y., Gong, P., Mayne, C. G., Srinivasan, S., Kim, S. H., Carlson, K. E., Nettles, K. W., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jul 27 2017, In : Journal of Medicinal Chemistry. 60, 14, p. 6321-6336 16 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Breast Neoplasms
Down-Regulation
Ligands
Adenoviridae
Estrogen Receptors
Estrogens
Cell Proliferation
Breast Neoplasms

Affinity Labeling of Receptors for Steroid and Thyroid Hormones

Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 1984, In : Vitamins and Hormones. 41, C, p. 213-281 69 p.

Research output: Contribution to journalArticle

Thyroid Hormone Receptors
Binding Sites
Molecular Probes
Proteins
Hormones

A human estrogen receptor (ER)α mutation with differential responsiveness to nonsteroidal ligands: Novel approaches for studying mechanism of ER action

Paulmurugan, R., Tamrazi, A., Katzenellenbogen, J. A., Katzenellenbogen, B. S. & Gambhir, S. S., Jul 1 2008, In : Molecular Endocrinology. 22, 7, p. 1552-1564 13 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Ligands
Mutation
Estradiol
Transcriptional Activation

Allosteric Control of Ligand Selectivity between Estrogen Receptors α and β: Implications for Other Nuclear Receptors

Nettles, K. W., Sun, J., Radek, J. T., Sheng, S., Rodriguez, A. L., Katzenellenbogen, J. A., Katzenellenbogen, B. S. & Greene, G. L., Feb 13 2004, In : Molecular cell. 13, 3, p. 317-327 11 p.

Research output: Contribution to journalArticle

Cytoplasmic and Nuclear Receptors
Estrogen Receptors
Ligands
Amino Acid Substitution
Signal Transduction
Estrogen Receptor Modulators
Tamoxifen
Protein Kinases
Breast Neoplasms
Cyclic AMP-Dependent Protein Kinases

Alteration of large-scale chromatin structure by estrogen receptor

Nye, A. C., Rajendran, R. R., Stenoien, D. L., Mancini, M. A., Katzenellenbogen, B. S. & Belmont, A. S., May 9 2002, In : Molecular and cellular biology. 22, 10, p. 3437-3449 13 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Chromatin
Lac Repressors
Estradiol
Nuclear Receptor Coactivator 1
Transforming Growth Factors
Estrogens
Steroids
Breast Neoplasms
Growth

Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open pocket conformation is required for ligand interaction

Carlson, K. E., Choi, I., Gee, A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 2 1997, In : Biochemistry. 36, 48, p. 14897-14905 9 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Conformations
Ligands
Estradiol
Association reactions
Mitogen-Activated Protein Kinase 1
Estrogen Receptors
Breast Neoplasms
MicroRNAs
Neoplasms

Analogs of methyl-piperidinopyrazole (MPP): Antiestrogens with estrogen receptor α selective activity

Zhou, H. B., Carlson, K. E., Stossi, F., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 1 2009, In : Bioorganic and Medicinal Chemistry Letters. 19, 1, p. 108-110 3 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Ether
Estrogens
Ligands

Analysis of estrogen receptor interaction with a repressor of estrogen receptor activity (REA) and the regulation of estrogen receptor transcriptional activity by REA

Delage-Mourroux, R., Martini, P. G. V., Choi, I., Kraichely, D. M., Hoeksema, J. & Katzenellenbogen, B. S., Nov 17 2000, In : Journal of Biological Chemistry. 275, 46, p. 35848-35856 9 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Competitive Binding
Response Elements
Cytoplasmic and Nuclear Receptors
Glutathione Transferase

Analysis of estrogen receptor transcriptional enhancement by a nuclear hormone receptor coactivator

Mcinerney, E. M., Tsai, M. J., O'Malley, B. W. & Katzenellenbogen, B. S., Sep 17 1996, In : Proceedings of the National Academy of Sciences of the United States of America. 93, 19, p. 10069-10073 5 p.

Research output: Contribution to journalArticle

Nuclear Receptor Coactivators
Cytoplasmic and Nuclear Receptors
Estrogen Receptors
Ligands
Nuclear Receptor Coactivator 1

Analysis of estrogen response element binding by genetically selected steroid receptor DNA binding domain mutants exhibiting altered specificity and enhanced affinity

Chusacultanachai, S., Glenn, K. A., Rodriguez, A. O., Read, E. K., Gardner, J. F., Katzenellenbogen, B. S. & Shapiro, D. J., Aug 13 1999, In : Journal of Biological Chemistry. 274, 33, p. 23591-23598 8 p.

Research output: Contribution to journalArticle

Steroid Receptors
Response Elements
Estrogens
Amino Acids
Bacteriophage P22

Analysis of mechanisms that determine dominant negative estrogen receptor effectiveness

Schodin, D. J., Zhuang, Y., Shapiro, D. J. & Katzenellenbogen, B. S., Dec 29 1995, In : Journal of Biological Chemistry. 270, 52, p. 31163-31171 9 p.

Research output: Contribution to journalArticle

Estrogen Receptors
Estrogens
Dimerization
Response Elements
Mutation
Bioactivity
Estrogen Receptors
Half-Life
Mutagenesis
Proteins
Estrogen Receptors
Dihydrotestosterone
Androgens
Proteins
Uterus
Androgen Antagonists
Androgen Receptors
Progesterone Receptors
Estrogen Receptors
Androgens

An efficient, general synthesis of alkylsulfinyltoluidides

Bowlus, S. B. & Katzenellenbogen, J. A., Jan 1 1974, In : Synthetic Communications. 4, 3, p. 137-141 5 p.

Research output: Contribution to journalArticle

An estrogen receptor-selective coregulator that potentiates the effectiveness of antiestrogens and represses the activity of estrogens

Montano, M. M., Ekena, K., Delage-Mourroux, R., Chang, W., Martini, P. & Katzenellenbogen, B. S., Jun 8 1999, In : Proceedings of the National Academy of Sciences of the United States of America. 96, 12, p. 6947-6952 6 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Estrogens
Cytoplasmic and Nuclear Receptors
Breast Neoplasms
Corpus Striatum
Estrogen Receptor Modulators
Dopamine Receptors
Spiperone
LY 117018
Eflornithine
Estrogen Receptor Modulators
Cell proliferation
Polyamines
Progesterone Receptors
Estrogen Receptor Modulators
Estrogen Receptors
Binding Sites
Growth
Tamoxifen
Estrogen Receptor Modulators
Progesterone Receptors
Growth and Development
Estrogen Receptors
9,10-Dimethyl-1,2-benzanthracene

Antagonists for Constitutively Active Mutant Estrogen Receptors: Insights into the Roles of Antiestrogen-Core and Side-Chain

Sharma, A., Toy, W., Guillen, V. S., Sharma, N., Min, J., Carlson, K. E., Mayne, C. G., Lin, S., Sabio, M., Greene, G., Katzenellenbogen, B. S., Chandarlapaty, S. & Katzenellenbogen, J. A., Dec 21 2018, In : ACS chemical biology. 13, 12, p. 3374-3384 11 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogen Receptors
Ligands
Cell proliferation
Breast Neoplasms

Antagonists selective for estrogen receptor α

Sun, J., Huang, Y. R., Harrington, W. R., Sheng, S., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 2002, In : Endocrinology. 143, 3, p. 941-947 7 p.

Research output: Contribution to journalArticle

Pyrazoles
Estrogen Receptor Modulators
Response Elements
Estrogens
Reporter Genes
Estrogen Receptor Modulators
Estrogen Receptors
Binding Sites
Cell Proliferation
Breast Neoplasms
Middle Hypothalamus
Estrogen Receptor Modulators
Prolactin
Dopamine
Estrogens

Antiestrogen action in the uterus: Biological ineffectiveness of nuclear bound estradiol after antiestrogen

Katzenellenbogen, B. S. & Ferguson, E. R., Jun 1975, In : Endocrinology. 97, 1, p. 1-12 12 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Uterus
Estradiol
Cytoplasmic and Nuclear Receptors
Weights and Measures
Estrogen Receptor Modulators
Tamoxifen
Estrogen Receptors
Estrogens
Estrogen Antagonists

Antiestrogen Binding in Antiestrogen Growth-resistant Estrogen-responsive Clonal Variants of MCF-7 Human Breast Cancer Cells

Miller, M. A., Lippman, M. E. & Katzenellenbogen, B. S., Nov 1 1984, In : Cancer Research. 44, 11, p. 5038-5045 8 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Estrogens
Estrogen Receptors
Breast Neoplasms
Growth
Estrogen Receptor Modulators
Tissue Distribution
Estrogen Receptors
Binding Sites
Ligands

Antiestrogenic Potency and Binding Characteristics of the Triphenylethylene H1285 in MCF-7 Human Breast Cancer Cells

Sheen, Y. Y., Ruh, T. S., Mangel, W. F. & Katzenellenbogen, B. S., Sep 1 1985, In : Cancer Research. 45, 9, p. 4192-4199 8 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Breast Neoplasms
Estrogen Receptors
Estradiol
Plasminogen Activators

Anti-estrogen interaction with uterine estrogen receptors. Studies with a radiolabeled anti-estrogen (CI-628)

Katzenellenbogen, B. S., Katzenellenbogen, J. A., Ferguson, E. R. & Krauthammer, N., Dec 1 1978, In : Journal of Biological Chemistry. 253, 3, p. 697-707 11 p.

Research output: Contribution to journalArticle

Nitromifene
Cytoplasmic and Nuclear Receptors
Estrogen Receptors
Estrogens
Sucrose

Antiestrogen Modulation of the Growth and Properties of Ovarian-Autonomous and Ovarian-Dependent Mammary Tumors in Rats

Tsai, T. L. S., Rutledge, S. & Katzenellenbogen, B. S., Dec 1 1979, In : Cancer Research. 39, 12, p. 5043-5050 8 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Breast Neoplasms
9,10-Dimethyl-1,2-benzanthracene
Growth
Ovariectomy

Antiestrogen pharmacology and mechanism of action

Katzenellenbogen, B. S., Miller, M. A., Eckert, R. L. & Sudo, K., Jan 1 1983, In : Journal of Steroid Biochemistry. 19, 1, p. 59-68 10 p.

Research output: Contribution to journalArticle

Estrogen Receptor Modulators
Pharmacology
Estrogen Receptors
Estrogens
Nuclear Proteins
Estrogen Receptor
Drug Resistance
Estrogen Receptor Modulators
Tamoxifen
Breast Cancer

Antiestrogens: Mechanisms of action and resistance in breast cancer

Katzenellenbogen, B. S., Montano, M. M., Ekena, K., Herman, M. E. & McInerney, E. M., Jan 1 1997, In : Breast Cancer Research and Treatment. 44, 1, p. 23-38 16 p.

Research output: Contribution to journalReview article

Estrogen Receptor Modulators
Estrogen Receptors
Breast Neoplasms
Estrogens
Hormones