Benita S Katzenellenbogen

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Research Output

1996

A transcriptionally active estrogen receptor mutant is a novel type of dominant negative inhibitor of estrogen action

McInerney, E. M., Ince, B. A., Shapiro, D. J. & Katzenellenbogen, B. S., Dec 17 1996, In : Molecular Endocrinology. 10, 12, p. 1519-1526 8 p.

Research output: Contribution to journalArticle

Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein

Weis, K. E., Ekena, K., Thomas, J. A., Lazennec, G. & Katzenellenbogen, B. S., Dec 1 1996, In : Molecular Endocrinology. 10, 11, p. 1388-1398 11 p.

Research output: Contribution to journalArticle

Estrogen receptors: Bioactivities and interactions with cell signaling pathways

Katzenellenbogen, B. S., Feb 1 1996, In : Biology of reproduction. 54, 2, p. 287-293 7 p.

Research output: Contribution to journalArticle

Identification of amino acids in the hormone binding domain of the human estrogen receptor important in estrogen binding

Ekena, K., Weis, K. E., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Sep 5 1996, In : Journal of Biological Chemistry. 271, 33, p. 20053-20059 7 p.

Research output: Contribution to journalArticle

Nuclear hormone receptors: Ligand-activated regulators of transcription and diverse cell responses

Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jul 1996, In : Chemistry and Biology. 3, 7, p. 529-536 8 p.

Research output: Contribution to journalReview article

Tripartite steroid hormone receptor pharmacology: Interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones

Katzenellenbogen, J. A., O'Malley, B. W. & Katzenellenbogen, B. S., Feb 13 1996, In : Molecular Endocrinology. 10, 2, p. 119-131 13 p.

Research output: Contribution to journalShort survey

1997

17α-(Haloacetamidoalkyl)estradiols alkylate the human estrogen receptor at cysteine residues 417 and 530

Aliau, S., El Garrouj, D., Yasri, A., Katzenellenbogen, B. S. & Borgna, J. L., May 13 1997, In : Biochemistry. 36, 19, p. 58615867 1 p.

Research output: Contribution to journalArticle

Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open pocket conformation is required for ligand interaction

Carlson, K. E., Choi, I., Gee, A., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 2 1997, In : Biochemistry. 36, 48, p. 14897-14905 9 p.

Research output: Contribution to journalArticle

Antiestrogens: Mechanisms of action and resistance in breast cancer

Katzenellenbogen, B. S., Montano, M. M., Ekena, K., Herman, M. E. & McInerney, E. M., Jan 1 1997, In : Breast Cancer Research and Treatment. 44, 1, p. 23-38 16 p.

Research output: Contribution to journalReview article

Different residues of the human estrogen receptor are involved in the recognition of structurally diverse estrogens and antiestrogens

Ekena, K., Weise, K. E., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Feb 21 1997, In : Journal of Biological Chemistry. 272, 8, p. 5069-5075 7 p.

Research output: Contribution to journalArticle

Editorial: A new actor in the estrogen receptor drama - Enter ER-β

Katzenellenbogen, B. S. & Korach, K. S., Jan 1 1997, In : Endocrinology. 138, 3, p. 861-862 2 p.

Research output: Contribution to journalEditorial

1998

Determinants of ligand specificity of estrogen receptor-α: Estrogen versus androgen discrimination

Ekena, K., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 9 1998, In : Journal of Biological Chemistry. 273, 2, p. 693-699 7 p.

Research output: Contribution to journalArticle

Estrogen receptor activation function 1 works by binding p160 coactivator proteins

Webb, P., Nguyen, P., Shinsako, J., Anderson, C., Feng, W., Nguyen, M. P., Chen, D., Huang, S. M., Subramanian, S., McKinerney, E., Katzenellenbogen, B. S., Stallcup, M. R. & Kushner, P. J., Jan 1 1998, In : Molecular Endocrinology. 12, 10, p. 1605-1618 14 p.

Research output: Contribution to journalArticle

Transcription activation by the human estrogen receptor subtype β (ERβ) studied with ERβ and ERα receptor chimeras

Mcinerney, E. M., Weis, K. E., Sun, J., Mosselman, S. & Katzenellenbogen, B. S., Jan 1 1998, In : Endocrinology. 139, 11, p. 4513-4522 10 p.

Research output: Contribution to journalArticle

Transcriptional regulation of the human quinone reductase gene by antiestrogen-liganded estrogen receptor-α and estrogen receptor-β

Montano, M. M., Jaiswal, A. K. & Katzenellenbogen, B. S., Sep 25 1998, In : Journal of Biological Chemistry. 273, 39, p. 25443-25449 7 p.

Research output: Contribution to journalArticle

1999

Analysis of estrogen response element binding by genetically selected steroid receptor DNA binding domain mutants exhibiting altered specificity and enhanced affinity

Chusacultanachai, S., Glenn, K. A., Rodriguez, A. O., Read, E. K., Gardner, J. F., Katzenellenbogen, B. S. & Shapiro, D. J., Aug 13 1999, In : Journal of Biological Chemistry. 274, 33, p. 23591-23598 8 p.

Research output: Contribution to journalArticle

An estrogen receptor-selective coregulator that potentiates the effectiveness of antiestrogens and represses the activity of estrogens

Montano, M. M., Ekena, K., Delage-Mourroux, R., Chang, W., Martini, P. & Katzenellenbogen, B. S., Jun 8 1999, In : Proceedings of the National Academy of Sciences of the United States of America. 96, 12, p. 6947-6952 6 p.

Research output: Contribution to journalArticle

Caveolin-1 potentiates estrogen receptor α (ERα) signaling. Caveolin-1 drives ligand-independent nuclear translocation and activation of ERα

Schlegel, A., Wang, C., Katzenellenbogen, B. S., Pestell, R. G. & Lisanti, M. P., Nov 19 1999, In : Journal of Biological Chemistry. 274, 47, p. 33551-33556 6 p.

Research output: Contribution to journalArticle

Coactivator peptides have a differential stabilizing effect on the binding of Estrogens and Antiestrogens with the estrogen receptor

Gee, A. C., Carlson, K. E., Martini, P. G. V., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jan 1 1999, In : Molecular Endocrinology. 13, 11, p. 1912-1923 12 p.

Research output: Contribution to journalArticle

Estrogen receptor regulation of the Na+/H+ exchanger regulatory factor

Ediger, T. R., Kraus, W. L., Weinman, E. J. & Katzenellenbogen, B. S., Jan 1 1999, In : Endocrinology. 140, 7, p. 2976-2982 7 p.

Research output: Contribution to journalArticle

Estrogen receptor subtype-selective ligands: Asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl-5,6,11,12- tetrahydrochrysenes

Meyers, M. J., Jun, S., Carlson, K. E., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jul 1 1999, In : Journal of Medicinal Chemistry. 42, 13, p. 2456-2468 13 p.

Research output: Contribution to journalArticle

Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-α or estrogen receptor-β

Sun, J., Meyers, M. J., Fink, B. E., Rajendran, R., Katzenellenbogen, J. A. & Katzenellenbogen, B. S., Jan 1 1999, In : Endocrinology. 140, 2, p. 800-804 5 p.

Research output: Contribution to journalArticle

The estrogen receptor enhances AP-1 activity by two distinct mechanisms with different requirements for receptor transactivation functions

Webb, P., Nguyen, P., Valentine, C., Lopez, G. N., Kwok, G. R., McInerney, E., Katzenellenbogen, B. S., Enmark, E., Gustafsson, J. Å., Nilsson, S. & Kushner, P. J., Jan 1 1999, In : Molecular Endocrinology. 13, 10, p. 1672-1685 14 p.

Research output: Contribution to journalArticle

2000

Activation of estrogen receptor-α by the heavy metal cadmium

Stoica, A., Katzenellenbogen, B. S. & Martin, M. B., Dec 1 2000, In : Molecular Endocrinology. 14, 4, p. 545-553 9 p.

Research output: Contribution to journalArticle

Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction

Stauffer, S. R., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Jun 1 2000, In : Bioorganic and Medicinal Chemistry. 8, 6, p. 1293-1316 24 p.

Research output: Contribution to journalArticle

Analysis of estrogen receptor interaction with a repressor of estrogen receptor activity (REA) and the regulation of estrogen receptor transcriptional activity by REA

Delage-Mourroux, R., Martini, P. G. V., Choi, I., Kraichely, D. M., Hoeksema, J. & Katzenellenbogen, B. S., Nov 17 2000, In : Journal of Biological Chemistry. 275, 46, p. 35848-35856 9 p.

Research output: Contribution to journalArticle

A role for Akt in mediating the estrogenic functions of epidermal growth factor and insulin-like growth factor I

Martin, M. B., Franke, T. F., Stoica, G. E., Chambon, P., Katzenellenbogen, B. S., Stoica, B. A., McLemore, M. S., Olivo, S. E. & Stoica, A., Jan 1 2000, In : Endocrinology. 141, 12, p. 4503-4511 9 p.

Research output: Contribution to journalArticle

Estrogen receptor alpha and estrogen receptor beta: Regulation by selective estrogen receptor modulators and importance in breast cancer

Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 1 2000, In : Breast Cancer Research. 2, 5, p. 335-344 10 p.

Research output: Contribution to journalReview article

Estrogen receptor-KRAB chimeras are potent ligand-dependent repressors of estrogen-regulated gene expression

De Haan, G., Chusacultanachai, S., Mao, C., Katzenellenbogen, B. S. & Shapiro, D. J., May 5 2000, In : Journal of Biological Chemistry. 275, 18, p. 13493-13501 9 p.

Research output: Contribution to journalArticle

Estrogen receptors: Selective ligands, partners, and distinctive pharmacology

Katzenellenbogen, B. S., Montano, M. M., Ediger, T. R., Sun, J., Ekena, K., Lazennec, G., Martini, P. G. V., McInerney, E. M., Delage-Mourroux, R., Weis, K., Katzenellenbogen, J. A., Nagel, S., Schrader, W., Bethea, C., Cutler, G. & Hock, J., Dec 1 2000, In : Recent Progress in Hormone Research. 55, p. 163-195 33 p.

Research output: Contribution to journalArticle

Molecular mechanisms of estrogen action: Selective ligands and receptor pharmacology

Katzenellenbogen, B. S., Choi, I., Delage-Mourroux, R., Ediger, T. R., Martini, P. G. V., Montano, M., Sun, J., Weis, K. & Katzenellenbogen, J. A., Nov 30 2000, In : Journal of Steroid Biochemistry and Molecular Biology. 74, 5, p. 279-285 7 p.

Research output: Contribution to journalArticle

Multistep signaling and transcriptional requirements for pituitary organogenesis in vivo

Rosenfeld, M. G., Briata, P., Dasen, J., Gleiberman, A. S., Kioussi, C., Lin, C., O'Connell, S. M., Ryan, A., Szeto, D. P., Treier, M., Katzenellenbogen, B., Nilson, J., Lawrence, A., Arnhold, I., Frohman, L. & Kochupillai, N., Dec 1 2000, In : Recent Progress in Hormone Research. 55, p. 1-14 14 p.

Research output: Contribution to journalArticle

Prothymosin alpha selectively enhances estrogen receptor transcriptional activity by interacting with a repressor of estrogen receptor activity

Martini, P. G. V., Delage-Mourroux, R., Kraichely, D. M. & Katzenellenbogen, B. S., Sep 6 2000, In : Molecular and cellular biology. 20, 17, p. 6224-6232 9 p.

Research output: Contribution to journalArticle

Pyrazole ligands: Structure - Affinity/activity relationships and estrogen receptor-α-selective agonists

Stauffer, S. R., Coletta, C. J., Tedesco, R., Nishiguchi, G., Carlson, K., Sun, J., Katzenellenbogen, B. S. & Katzenellenbogen, J. A., Dec 28 2000, In : Journal of Medicinal Chemistry. 43, 26, p. 4934-4947 14 p.

Research output: Contribution to journalArticle

2001

Activation of estrogen receptor β is a prerequisite for estrogen-dependent upregulation of nitric oxide synthases in neonatal rat cardiac myocytes

Nuedling, S., Karas, R. H., Mendelsohn, M. E., Katzenellenbogen, J. A., Katzenellenbogen, B. S., Meyer, R., Vetter, H. & Grohé, C., Aug 3 2001, In : FEBS Letters. 502, 3, p. 103-108 6 p.

Research output: Contribution to journalArticle

Direct Acetylation of the Estrogen Receptor α Hinge Region by p300 Regulates Transactivation and Hormone Sensitivity

Wang, C., Fu, M., Angeletti, R. H., Siconolfi-Baez, L., Reutens, A. T., Albanese, C., Lisanti, M. P., Katzenellenbogen, B. S., Kato, S., Hopp, T., Fuqua, S. A. W., Lopez, G. N., Kushner, P. J. & Pestell, R. G., Jan 25 2001, In : Journal of Biological Chemistry. 276, 21, p. 18375-18383 9 p.

Research output: Contribution to journalArticle